Interleukin-6 trans signalling enhances photodynamic therapy by modulating cell cycling

Br J Cancer. 2007 Dec 3;97(11):1513-22. doi: 10.1038/sj.bjc.6604073. Epub 2007 Nov 6.

Abstract

Photodynamic therapy (PDT) of solid tumours causes tissue damage that elicits local and systemic inflammation with major involvement of interleukin-6 (IL-6). We have previously reported that PDT-treated cells lose responsiveness to IL-6 cytokines. Therefore, it is unclear whether PDT surviving tumour cells are subject to regulation by IL-6 and whether this regulation could contribute to tumour control by PDT. We demonstrate in epithelial tumour cells that while the action of IL-6 cytokines through their membrane receptors is attenuated, regulation by IL-6 via trans-signalling is established. Soluble interleukin-6 receptor-alpha (IL-6Ralpha) (sIL-6Ralpha) and IL-6 were released by leucocytes in the presence of conditioned medium from PDT-treated tumour cells. Cells that had lost their membrane receptor IL-6Ralpha due to PDT responded to treatment with the IL-6R-IL-6 complex (Hyper-IL-6) with activation of signal transducers and activator of transcription (STAT3) and ERK. Photodynamic therapy-treated cells, which were maintained during post-PDT recovery in presence of IL-6 or Hyper-IL-6, showed an enhanced suppression of proliferation. Cytokine-dependent inhibition of proliferation correlated with a decrease in cyclin E, CDK2 and Cdc25A, and enhancement of p27kip1 and hypophosphorylated Rb. The IL-6 trans-signalling-mediated attenuation of cell proliferation was also effective in vivo detectable by an improved Colon26 tumour cure by PDT combined with Hyper-IL-6 treatment. Prevention of IL-6 trans-signalling using soluble gp130 reduced curability. The data suggest that the post-PDT tumour milieu contains the necessary components to establish effective IL-6 trans-signalling, thus providing a means for more effective tumour control.

MeSH terms

  • Animals
  • Blotting, Western
  • Cell Cycle / drug effects
  • Cell Cycle / physiology*
  • Cell Line, Tumor
  • Cell Proliferation / drug effects
  • Chlorophyll / analogs & derivatives
  • Chlorophyll / pharmacology
  • Colonic Neoplasms / metabolism
  • Colonic Neoplasms / pathology
  • Culture Media, Conditioned / pharmacology
  • Cyclin E / metabolism
  • Cyclin-Dependent Kinase 2 / metabolism
  • Cyclin-Dependent Kinase Inhibitor p27 / metabolism
  • Dose-Response Relationship, Drug
  • HeLa Cells
  • Humans
  • Interleukin-6 / metabolism
  • Interleukin-6 / pharmacology
  • Interleukin-6 / physiology*
  • Macrophages / drug effects
  • Macrophages / metabolism
  • Mice
  • Mice, Inbred BALB C
  • Photochemotherapy
  • Receptors, Interleukin-6 / metabolism
  • STAT3 Transcription Factor / metabolism
  • Signal Transduction / physiology*
  • cdc25 Phosphatases / metabolism

Substances

  • Culture Media, Conditioned
  • Cyclin E
  • Interleukin-6
  • Receptors, Interleukin-6
  • STAT3 Transcription Factor
  • interleukin-6 receptor alpha
  • Chlorophyll
  • Cyclin-Dependent Kinase Inhibitor p27
  • 2-(1-hexyloxyethyl)-2-devinyl pyropheophorbide-a
  • Cyclin-Dependent Kinase 2
  • cdc25 Phosphatases