[In vitro methods suitable for the prediction of drug and ABC transporter, especially ABCG2 interactions]

Acta Pharm Hung. 2007;77(4):205-16.
[Article in Hungarian]

Abstract

ABCG2, a transporter of the ATP-binding cassette family, is known to play a prominent role in the absorption, distribution, metabolism, and excretion of xenobiotics. Drug-transporter interactions are commonly screened by in vitro systems using transfected insect and/or human cell lines.

MeSH terms

  • ATP Binding Cassette Transporter, Subfamily G, Member 2
  • ATP-Binding Cassette Transporters / drug effects
  • ATP-Binding Cassette Transporters / metabolism*
  • Animals
  • Biological Transport
  • Cell Line
  • Drug Interactions
  • Drug Therapy
  • Humans
  • Insecta
  • Neoplasm Proteins / drug effects
  • Neoplasm Proteins / metabolism*
  • Xenobiotics / pharmacokinetics

Substances

  • ABCG2 protein, human
  • ATP Binding Cassette Transporter, Subfamily G, Member 2
  • ATP-Binding Cassette Transporters
  • Neoplasm Proteins
  • Xenobiotics