Progestogens: therapeutic and adverse effects in early post-menopausal women

Maturitas. 1991 Mar;13(1):7-16. doi: 10.1016/0378-5122(91)90280-4.

Abstract

Progestogen treatment is associated with a number of subjective symptoms. In the present study, 148 healthy post-menopausal women suffering from mild climacteric symptoms were randomly allocated to 12 weeks of treatment with (a) 2 mg oestradiol valerate combined with cyproterone acetate, medroxyprogesterone acetate or levonorgestrel; (b) 1.5 mg 17 beta-oestradiol combined with desogestrel; or (c) placebo. Climacteric symptoms, Kupperman index scores and potential adverse progestogen effects were recorded before treatment and three times per month during therapy. All the hormone regimens had a rapid effect, reducing the severity of climacteric symptoms to about 30% of the baseline values (P less than 0.001) within one month. Hot flushes were reduced in severity and/or frequency by 76 100% within 3 months (P less than 0.001). The regimens which included hydroxyprogesterone derivatives produced a transient increase in breast tenderness. Other recorded potential adverse progestogen effects showed no significant changes during the study. We concluded that the addition of progestogens (whether 19-nortestosterone or hydroxyprogesterone derivatives) does not produce significant side effects during combined hormone replacement therapy.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial

MeSH terms

  • Androgen Antagonists / administration & dosage
  • Androgen Antagonists / adverse effects
  • Androgen Antagonists / therapeutic use*
  • Climacteric / blood
  • Climacteric / drug effects*
  • Climacteric / physiology
  • Cyproterone / administration & dosage
  • Cyproterone / adverse effects
  • Cyproterone / analogs & derivatives*
  • Cyproterone / therapeutic use
  • Cyproterone Acetate
  • Drug Therapy, Combination
  • Estradiol / administration & dosage
  • Estradiol / adverse effects
  • Estradiol / analogs & derivatives*
  • Estradiol / blood
  • Estradiol / therapeutic use
  • Female
  • Humans
  • Levonorgestrel
  • Medroxyprogesterone / administration & dosage
  • Medroxyprogesterone / adverse effects
  • Medroxyprogesterone / therapeutic use*
  • Middle Aged
  • Norgestrel / administration & dosage
  • Norgestrel / adverse effects
  • Norgestrel / therapeutic use*
  • Severity of Illness Index

Substances

  • Androgen Antagonists
  • Norgestrel
  • Cyproterone Acetate
  • Estradiol
  • Levonorgestrel
  • Cyproterone
  • Medroxyprogesterone