Prothrombotic effect of Rofecoxib in a murine venous thrombosis model

Thromb Res. 2008;122(5):668-73. doi: 10.1016/j.thromres.2008.04.016. Epub 2008 Jun 20.

Abstract

The potential prothrombotic effect of the cyclooxygenase-2 (COX-2) inhibitor Rofecoxib (Vioxx) was investigated using murine thrombosis models. In a jugular vein thrombosis model (photochemically induced injury) in lean wild-type mice, Rofecoxib treatment for 4 weeks induced a mild prothrombotic tendency, as indicated by a shorter occlusion time as compared to placebo (median of 12 min versus 36 min; p < 0.05). Thrombus size was somewhat, but not significantly, enhanced after Rofecoxib treatment. In a femoral artery thrombosis model (FeCl3 induced injury) Rofecoxib did not cause an enhanced thrombotic tendency in mice with nutritionally induced or genetically determined (ob/ob) obesity. The occlusion time was comparable for obese wild-type mice with (8.8+/-0.7 min) or without (7.8+/-2.1 min) Rofecoxib treatment, as well as for ob/ob mice (8.5+/-0.7 min versus 6.8+/-3.0 min). Thus, an enhanced prothrombotic effect of Rofecoxib was detected when using a venous thrombosis model in lean mice, but not when using an arterial thrombosis model in obese mice.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cyclooxygenase 2 Inhibitors / toxicity*
  • Disease Models, Animal
  • Femoral Artery
  • Jugular Veins
  • Lactones / toxicity*
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Mice, Obese
  • Obesity / blood
  • Obesity / complications
  • Platelet Aggregation / drug effects
  • Sulfones / toxicity*
  • Thrombosis / blood
  • Thrombosis / chemically induced
  • Thrombosis / etiology
  • Venous Thrombosis / blood
  • Venous Thrombosis / chemically induced*
  • Venous Thrombosis / etiology

Substances

  • Cyclooxygenase 2 Inhibitors
  • Lactones
  • Sulfones
  • rofecoxib