Mitogen-activated protein kinase p38 pathway in venous ulcer fibroblasts

Vasc Endovascular Surg. 2008 Aug-Sep;42(4):367-74. doi: 10.1177/1538574408316140. Epub 2008 Jun 25.

Abstract

Objective: Venous ulcer fibroblasts (w-fb) have attenuated growth compared to normal fibroblasts (n-fb). The MAPKp38 pathway mediates stress-responses in various diseases. We hypothesize that p38 pathway is altered in w-fb.

Methods: W-fb were isolated from venous ulcers and n-fb from the ipsilateral thigh. Fibroblasts were analyzed for phosphorylated p38 using immunoblot. The relation between p38 and w-fb proliferation was assessed with SB203580 (p38 inhibitor). Fibroblasts were treated with bFGF, TNF-a, and IL-1 and p38 expression analyzed.

Results: Phosphorylated p38 expression was increased in w-fb (AU%=233.5+/-59.7, P=0.039) compared to n-fb (AU%=99.9+/-14.6). W-fb treated with SB203580 demonstrated increased growth compared to untreated w-fb. W-fb treated with bFGF demonstrated decreased p38. TNF-alpha and IL-1beta significantly increase p38 expression.

Conclusions: MAPK p38 is up-regulated in w-fb. Regulation of w-fb proliferation is influenced by p38. Altering the p38 pathway in vivo with growth factors or cytokine inhibition may improve fibroblast proliferation and venous ulcer healing.

MeSH terms

  • Adult
  • Aged
  • Cell Proliferation* / drug effects
  • Cells, Cultured
  • Female
  • Fibroblast Growth Factor 2 / metabolism
  • Fibroblasts / drug effects
  • Fibroblasts / enzymology*
  • Fibroblasts / pathology
  • Humans
  • Imidazoles / pharmacology
  • Interleukin-1 / metabolism
  • Male
  • Middle Aged
  • Phosphorylation
  • Protein Kinase Inhibitors / pharmacology
  • Pyridines / pharmacology
  • Tumor Necrosis Factor-alpha / metabolism
  • Up-Regulation
  • Varicose Ulcer / enzymology*
  • Varicose Ulcer / pathology
  • p38 Mitogen-Activated Protein Kinases / antagonists & inhibitors
  • p38 Mitogen-Activated Protein Kinases / metabolism*

Substances

  • Imidazoles
  • Interleukin-1
  • Protein Kinase Inhibitors
  • Pyridines
  • Tumor Necrosis Factor-alpha
  • Fibroblast Growth Factor 2
  • p38 Mitogen-Activated Protein Kinases
  • SB 203580