Copper-catalyzed sonogashira-type reactions under mild palladium-free conditions

Org Lett. 2008 Aug 7;10(15):3203-6. doi: 10.1021/ol801025u. Epub 2008 Jun 28.

Abstract

We have developed an inexpensive catalytic system using a readily available copper/ligand combination for the Sonogashira-type cross-coupling of aryl iodides and phenyl- and hexyl-acetylene which affords disubstituted alkynes in good to excellent yields.