Usefulness of a selective neutrophil elastase inhibitor (sivelestat) in septic ARDS patients after gastrointestinal surgery

Hepatogastroenterology. 2008 May-Jun;55(84):967-73.

Abstract

Background/aims: The usefulness of a neutrophil elastase inhibitor (sivelestat) was evaluated for treating septic acute respiratory distress syndrome (ARDS) after gastrointestinal surgery.

Methodology: The subjects were 36 patients with septic ARDS after gastrointestinal surgery. ARDS was defined as acute lung injury associated with systemic inflammatory response syndrome. Sivelestat was intravenously administered at a dose of 0.2 mg/kg/hr continuously for 3 days or more. The effectiveness of sivelestat was evaluated based on the lung injury score, P/F ratio, and ventilator free days (VFD).

Results: Marked responses were observed in 12 patients (33.3%), responses in 17 (47.2%), and no response in 7 (19.4%). In the patients with marked responses or responses (responders), the P/F ratio was significantly improved on day 3 of drug administration and at the end of administration compared with the pre-administration ratio. Comparison between the responders and non-responders showed significant differences on day 3 and at the end of drug administration. VFD significantly differed between the responders (18.8 days) and the non-responders (11.0 days).

Conclusion: In conclusion, sivelestat may be effective against septic ARDS. The effectiveness of the drug could be determined based on improvement in oxygenation ability on day 3 of drug administration.

MeSH terms

  • Acute Lung Injury / drug therapy*
  • Acute Lung Injury / etiology
  • Adult
  • Aged
  • Critical Care
  • Drug Administration Schedule
  • Female
  • Gastrointestinal Neoplasms / surgery*
  • Glycine / analogs & derivatives*
  • Glycine / therapeutic use
  • Humans
  • Infusions, Intravenous
  • Leukocyte Elastase / antagonists & inhibitors*
  • Male
  • Middle Aged
  • Oxygen / blood
  • Positive-Pressure Respiration
  • Postoperative Complications / drug therapy*
  • Postoperative Complications / etiology
  • Respiratory Distress Syndrome / drug therapy*
  • Respiratory Distress Syndrome / etiology
  • Sepsis / drug therapy*
  • Serine Proteinase Inhibitors / therapeutic use*
  • Sulfonamides / therapeutic use*
  • Systemic Inflammatory Response Syndrome / drug therapy*
  • Systemic Inflammatory Response Syndrome / etiology

Substances

  • Serine Proteinase Inhibitors
  • Sulfonamides
  • sivelestat
  • Leukocyte Elastase
  • Oxygen
  • Glycine