Involvement of endothelin-1 in habitual exercise-induced increase in arterial compliance

Acta Physiol (Oxf). 2009 Jun;196(2):223-9. doi: 10.1111/j.1748-1716.2008.01909.x. Epub 2008 Oct 4.

Abstract

Aim: Habitual aerobic exercise results in a significant increase in central arterial compliance. Endothelin-1 (ET-1) is a potent endothelium-derived vasoconstrictor peptide and could play a role in mediating the habitual aerobic exercise-induced increase in central arterial compliance. The aim of the present study was to examine whether ET-1 is involved in the mechanisms underlying the increase in central arterial compliance with aerobic exercise training.

Methods: Seven apparently healthy middle-aged and older (60 +/- 3 years) adults underwent systemic endothelin-A/B (ET(A/B))-receptor blockade (500 mg of Tracleer) before and after 12 weeks of aerobic exercise training (70 +/- 1% of maximal heart rate, 44 +/- 2 min day(-1), 4.4 +/- 0.1 days week(-1)).

Results: Basal carotid arterial compliance (via simultaneous B-mode ultrasound and arterial applanation tonometry on the common carotid artery) increased significantly after exercise training. Resting plasma ET-1 concentration decreased significantly after exercise training. Before exercise intervention, carotid arterial compliance increased significantly with the administration of the ET(A/B)-receptor blockade. After training, however, increases in carotid arterial compliance previously observed with the ET(A/B)-receptor blockade before training were abolished.

Conclusions: Regular aerobic exercise training enhances central arterial compliance in middle-aged and older humans. The increase in arterial compliance was associated with the corresponding reduction in plasma ET-1 concentration as well as the elimination of ET-1-mediated vascular tone. These results suggest that reductions in ET-1 may be an important mechanism underlying the beneficial effect of exercise training on central artery compliance.

Publication types

  • Clinical Trial
  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adipose Tissue / physiology
  • Aged
  • Antihypertensive Agents / pharmacology
  • Arteries / anatomy & histology
  • Arteries / drug effects
  • Arteries / physiology*
  • Blood Glucose / physiology
  • Blood Pressure / drug effects
  • Blood Pressure / physiology
  • Body Weight / physiology
  • Bosentan
  • Carotid Arteries / anatomy & histology
  • Cholesterol / blood
  • Compliance / drug effects
  • Compliance / physiology
  • Endothelin Receptor Antagonists
  • Endothelin-1 / antagonists & inhibitors
  • Endothelin-1 / blood*
  • Exercise / physiology*
  • Female
  • Heart Rate / drug effects
  • Heart Rate / physiology
  • Humans
  • Male
  • Middle Aged
  • Sulfonamides / pharmacology

Substances

  • Antihypertensive Agents
  • Blood Glucose
  • Endothelin Receptor Antagonists
  • Endothelin-1
  • Sulfonamides
  • Cholesterol
  • Bosentan