C-terminal ADAMTS-18 fragment induces oxidative platelet fragmentation, dissolves platelet aggregates, and protects against carotid artery occlusion and cerebral stroke

Blood. 2009 Jun 11;113(24):6051-60. doi: 10.1182/blood-2008-07-170571. Epub 2009 Feb 13.

Abstract

Anti-platelet integrin GPIIIa49-66 antibody (Ab) induces complement-independent platelet oxidative fragmentation and death by generation of platelet peroxide following NADPH oxidase activation. A C-terminal 385-amino acid fragment of ADAMTS-18 (a disintegrin metalloproteinase with thrombospondin motifs produced in endothelial cells) induces oxidative platelet fragmentation in an identical kinetic fashion as anti-GPIIIa49-66 Ab. Endothelial cell ADAMTS-18 secretion is enhanced by thrombin and activated by thrombin cleavage to fragment platelets. Platelet aggregates produced ex vivo with ADP or collagen and fibrinogen are destroyed by the C-terminal ADAMTS-18 fragment. Anti-ADAMTS-18 Ab shortens the tail vein bleeding time. The C-terminal fragment protects against FeCI3-induced carotid artery thrombosis as well as cerebral infarction in a postischemic stroke model. Thus, a new mechanism is proposed for platelet thrombus clearance, via platelet oxidative fragmentation induced by thrombin cleavage of ADAMTS-18.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • ADAM Proteins / metabolism
  • ADAM Proteins / pharmacology*
  • ADAMTS Proteins
  • Animals
  • Bleeding Time
  • Blood Platelets / metabolism*
  • Blood Platelets / pathology
  • Carotid Stenosis / metabolism
  • Carotid Stenosis / pathology
  • Carotid Stenosis / prevention & control*
  • Cyclic AMP / pharmacology
  • Endothelium, Vascular / metabolism
  • Humans
  • Immunoenzyme Techniques
  • Mice
  • Mice, Inbred BALB C
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Peptide Fragments / pharmacology*
  • Peptide Library
  • Platelet Aggregation / drug effects*
  • Platelet Glycoprotein GPIIb-IIIa Complex / pharmacology
  • Polymerase Chain Reaction
  • Stroke / metabolism
  • Stroke / pathology
  • Stroke / prevention & control*
  • Thrombin / pharmacology
  • Umbilical Veins / cytology

Substances

  • Peptide Fragments
  • Peptide Library
  • Platelet Glycoprotein GPIIb-IIIa Complex
  • platelet glycoprotein (GP)IIIa 49-66
  • Cyclic AMP
  • Thrombin
  • ADAM Proteins
  • ADAMTS Proteins
  • ADAMTS18 protein, human