Smooth muscle archvillin is an ERK scaffolding protein

J Biol Chem. 2009 Jun 26;284(26):17607-15. doi: 10.1074/jbc.M109.002386. Epub 2009 Apr 29.

Abstract

ERK influences a number of pathways in all cells, but how ERK activities are segregated between different pathways has not been entirely clear. Using immunoprecipitation and pulldown experiments with domain-specific recombinant fragments, we show that smooth muscle archvillin (SmAV) binds ERK and members of the ERK signaling cascade in a domain-specific, stimulus-dependent, and pathway-specific manner. MEK binds specifically to the first 445 residues of SmAV. B-Raf, an upstream regulator of MEK, constitutively interacts with residues 1-445 and 446-1250. Both ERK and 14-3-3 bind to both fragments, but in a stimulus-specific manner. Phosphorylated ERK is associated only with residues 1-445. An ERK phosphorylation site was determined by mass spectrometry to reside at Ser132. A phospho-antibody raised to this site shows that the site is phosphorylated during alpha-agonist-mediated ERK activation in smooth muscle tissue. Phosphorylation of SmAV by ERK decreases the association of phospho-ERK with SmAV. These results, combined with previous observations, indicate that SmAV serves as a new ERK scaffolding protein and provide a mechanism for regulation of ERK binding, activation, and release from the signaling complex.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • 14-3-3 Proteins / metabolism
  • Amino Acid Sequence
  • Animals
  • Aorta / cytology
  • Aorta / metabolism
  • Ferrets
  • Immunoprecipitation
  • Mass Spectrometry
  • Membrane Proteins / metabolism*
  • Microfilament Proteins / metabolism*
  • Mitogen-Activated Protein Kinase 1 / metabolism*
  • Mitogen-Activated Protein Kinase 3 / metabolism*
  • Mitogen-Activated Protein Kinase Kinases / metabolism*
  • Molecular Sequence Data
  • Muscle, Smooth / cytology
  • Muscle, Smooth / metabolism*
  • Phosphorylation
  • Proto-Oncogene Proteins B-raf / metabolism
  • Signal Transduction

Substances

  • 14-3-3 Proteins
  • Membrane Proteins
  • Microfilament Proteins
  • BRAF protein, human
  • Proto-Oncogene Proteins B-raf
  • Mitogen-Activated Protein Kinase 1
  • Mitogen-Activated Protein Kinase 3
  • Mitogen-Activated Protein Kinase Kinases