Up-regulated microRNA-143 transcribed by nuclear factor kappa B enhances hepatocarcinoma metastasis by repressing fibronectin expression

Hepatology. 2009 Aug;50(2):490-9. doi: 10.1002/hep.23008.

Abstract

It is increasingly clear that hepatocellular carcinoma (HCC) has a distinct microRNA (miRNA) expression profile that is involved in malignancy; however, little is known about how functional miRNA modulates the metastasis of hepatitis B virus (HBV)-related HCC (HBV-HCC). In the present study, we demonstrate that the levels of miRNA-143 (miR-143) are dramatically increased in metastatic HBV-HCC of both p21-HBx transgenic mice and HCC patients. Moreover, we show that overexpression of this miRNA is transcribed by nuclear factor kappa B (NF-kappaB) and favors liver tumor cell invasive and metastatic behavior. Intratumoral administration of miR-143 shows that high levels of miR-143 can significantly promote HCC metastasis in an athymic nude mouse model. An in vivo study that used p21-HBx transgenic mice also showed that local liver metastasis and distant lung metastasis are significantly inhibited by blocking miR-143. Additionally, fibronectin type III domain containing 3B (FNDC3B), which regulates cell motility, was identified as the direct and functional target of miR-143 both in vivo and in vitro.

Conclusion: Up-regulation of miR-143 expression transcribed by NF-kappaB in HBV-HCC promotes cancer cell invasion/migration and tumor metastasis by repression of FNDC3B expression. The present study provides a better understanding of the specificity of the biological behavior and thus may be helpful in developing an effective treatment against HBV-HCC.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Aged
  • Animals
  • Carcinoma, Hepatocellular / metabolism*
  • Carcinoma, Hepatocellular / virology
  • Cell Line, Tumor
  • Cell Movement
  • Down-Regulation
  • Female
  • Fibronectins / metabolism*
  • Gene Expression Regulation, Neoplastic
  • Hepatitis B, Chronic / complications
  • Humans
  • Liver Neoplasms / metabolism*
  • Liver Neoplasms / virology
  • Male
  • Mice
  • Mice, Nude
  • Mice, Transgenic
  • MicroRNAs / metabolism*
  • Middle Aged
  • NF-kappa B / metabolism*
  • Neoplasm Invasiveness
  • Neoplasm Metastasis
  • Trans-Activators / genetics
  • Up-Regulation
  • Viral Regulatory and Accessory Proteins

Substances

  • FNDC3B protein, human
  • Fibronectins
  • MIRN143 microRNA, human
  • MicroRNAs
  • NF-kappa B
  • Trans-Activators
  • Viral Regulatory and Accessory Proteins
  • hepatitis B virus X protein