Palonosetron in prevention of nausea and vomiting after highly emetogenic chemotherapy before haematopoietic stem cell transplantation-single center experience

Transplant Proc. 2009 Oct;41(8):3247-9. doi: 10.1016/j.transproceed.2009.07.071.

Abstract

Objective: A clinical study of palonosetron was performed to evaluate its efficacy in preventing both acute and delayed emesis after high-dose chemotherapy (HDC) before hematopoietic stem cell transplantation (HSCT) using a historical control group of patients treated with ondansetron as the comparative drug.

Methods: Among the 46 evaluated patients 20 with lymphoma received BEAM as the conditioning regimen; 16 has relapsed germ cell tumors treated with CARBOPEC; and 10 with acute myeloid leukemia received BuCY. Increasing severity of nausea was evaluated according to the following 4-grade scale: none (no nausea); mild (slight nausea but no disruption to daily activities); moderate (nausea and some disruption to daily activities); and severe (extreme nausea and severe disruption to daily activities). The emetic response rate was evaluated using the criteria: complete (no emetic episode); major (1-2 episodes); minor (3-5 episodes); and failure (>5 episodes). The response rate of the study drugs was evaluated by the following 4-grade scale based on the condition of nausea and vomiting: highly effective, moderately effective, slightly effective, and not effective.

Results: Patients treated with palonosetron showed significantly greater response rates than those receiving ondansetron during the both the acute and the delayed phases: highly and moderately effective: acute phase 15% versus 5% CARBOPEC; 70% versus 35% BEAM and 32% versus 20% BuCY; delayed phase: 60% versus 30% BuCY; 100% versus 50% BEAM and 25% versus 10% CARBOPEC.

Conclusions: Single-dose palonosetron was more effective than ondansetron treatment to prevent acute and delayed nausea and vomiting following HDC before HSCT.

MeSH terms

  • Antineoplastic Agents / therapeutic use
  • Carmustine / therapeutic use
  • Emetics / adverse effects*
  • Emetics / therapeutic use*
  • Etoposide / therapeutic use
  • Hematopoietic Stem Cell Transplantation / adverse effects*
  • Humans
  • Isoquinolines / therapeutic use*
  • Lymphoma / drug therapy
  • Lymphoma / surgery
  • Nausea / prevention & control*
  • Ondansetron / therapeutic use
  • Palonosetron
  • Quinuclidines / therapeutic use*
  • Serotonin Antagonists / therapeutic use*
  • Treatment Outcome
  • Vomiting / prevention & control*

Substances

  • Antineoplastic Agents
  • Emetics
  • Isoquinolines
  • Quinuclidines
  • Serotonin Antagonists
  • Ondansetron
  • Palonosetron
  • Etoposide
  • Carmustine