Abstract
The peptide pyroGlu-Gln-Gly-Ser-Asn, recently isolated from mouse liver, inhibited DNA synthesis and proliferation in vitro of MH1C1 cells, a rat clonal strain derived from a Morris transplantable hepatoma. Both the biological peptide isolated from mouse liver and the synthetic homolog showed bell-shaped dose-response curves. Maximal inhibition (approximately 50%) was observed at two separate dose ranges: one at 10(-7)-10(-10) M, and one at 10(-14)-10(-15) M.
Publication types
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Research Support, Non-U.S. Gov't
MeSH terms
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Amino Acid Sequence
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Animals
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Cell Division / drug effects
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DNA / biosynthesis
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Dose-Response Relationship, Drug
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Liver / chemistry
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Liver / cytology
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Liver / drug effects*
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Liver / metabolism
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Liver Neoplasms, Experimental / drug therapy
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Liver Neoplasms, Experimental / pathology*
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Mice
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Molecular Sequence Data
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Neoplasm Transplantation
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Oligopeptides / pharmacology*
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Peptides / isolation & purification
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Peptides / pharmacology*
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Pyrrolidonecarboxylic Acid / analogs & derivatives
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Rats
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Time Factors
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Tumor Cells, Cultured
Substances
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Oligopeptides
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Peptides
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pyroglutamyl-glutaminyl-glycyl-seryl-asparagine
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DNA
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Pyrrolidonecarboxylic Acid