Signal transduction by interleukin 2 receptor beta chain: importance of the structural integrity as revealed by site-directed mutagenesis and generation of chimeric receptors

Int Immunol. 1991 Feb;3(2):149-56. doi: 10.1093/intimm/3.2.149.

Abstract

The functional interleukin 2 receptor (IL-2R) consists of at least two IL-2 binding cell surface molecules, IL-2R alpha and IL-2R beta, the latter component being responsible for the intracellular growth signal transduction. In this study we attempted to identify the critical amino acid residues in the cytoplasmic domain of human IL-2R beta for such signal transduction by expressing mutated IL-2R beta cDNAs in a pro-B cell line, BAF-B03. We demonstrate that a single amino acid substitution within the 'serine-rich' cytoplasmic region of IL-2R beta (i.e. Leu299 changed to Pro) completely abrogates the receptor function in growth stimulation, but not in ligand binding. We also show that the murine erythropoietin receptor (EPO-R) is functional in BAF-B03, but that chimeric receptors, essentially possessing the IL-2R beta extracellular and a homologous region derived from EPO-R cytoplasmic domain, are not capable of transducing the IL-2-induced signal.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • B-Lymphocytes / immunology
  • Base Sequence
  • Chimera / genetics*
  • Erythropoietin / genetics
  • Gene Expression
  • Humans
  • Interleukin-2 / metabolism
  • Molecular Sequence Data
  • Mutagenesis, Site-Directed / genetics*
  • Plasmids
  • Receptors, Interleukin-2 / genetics*
  • Sequence Homology, Nucleic Acid
  • Signal Transduction*
  • Structure-Activity Relationship
  • Transfection

Substances

  • Interleukin-2
  • Receptors, Interleukin-2
  • Erythropoietin