Modulation of E-cadherin expression by K-Ras; involvement of DNA methyltransferase-3b

Carcinogenesis. 2010 Jul;31(7):1194-201. doi: 10.1093/carcin/bgq071. Epub 2010 Apr 7.

Abstract

E-cadherin, as a tumor suppressor, plays an important role for intercellular adhesion involved in metastasis. Although K-Ras is highly expressed in a variety of cancers, the regulation of E-cadherin expression by K-Ras in association with DNA methylation and cell metastasis has not been completely clarified. In this study, E-cadherin expression was repressed in 267B1/K-Ras human epithelial prostate cancer cells stably overexpressing K-Ras, resulting from hypermethylation of E-cadherin promoter as evidenced by methylation-specific polymerase chain reaction (PCR), bisulfite sequencing, real-time reverse transcription-PCR and western blot analysis. The increased level of DNA methyltransferase (DNMT) 3b in 267B1/K-Ras cells was reduced by small interfering RNA-mediated knockdown of k-ras, whereas DNMT1 and DNMT3a did not change regardless of K-Ras or 5-aza-2'-deoxycytidine (5'-AzaC) treatment. Furthermore, binding of DNMT3b to E-cadherin promoter was increased in 267B1/K-Ras cells but was reduced by 5'-AzaC, as revealed by chromatin immunoprecipitation assay, which was in agreement with cell aggregation and invasive mobilization of the cells. Hence, our data suggest that increased binding of DNMT3b to E-cadherin promoter region by K-Ras cause promoter hypermethylation for reduced expression of E-cadherin, leading to the decreased cell aggregation and increased metastasis of human prostate cancer cells overexpressing K-Ras.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Azacitidine / analogs & derivatives
  • Azacitidine / pharmacology
  • Cadherins / genetics*
  • Cell Communication
  • Cell Line, Tumor
  • Cell Movement
  • CpG Islands
  • DNA (Cytosine-5-)-Methyltransferases / genetics
  • DNA (Cytosine-5-)-Methyltransferases / physiology*
  • DNA Methylation
  • DNA Methyltransferase 3B
  • Decitabine
  • Genes, ras*
  • Humans
  • Male
  • Promoter Regions, Genetic
  • Prostatic Neoplasms / pathology*

Substances

  • Cadherins
  • Decitabine
  • DNA (Cytosine-5-)-Methyltransferases
  • Azacitidine