Biomimetic construction of the hydroquinoline ring system. Diastereodivergent enantioselective synthesis of 2,5-disubstituted cis-decahydroquinolines

J Org Chem. 2010 Jun 4;75(11):3797-805. doi: 10.1021/jo1005894.

Abstract

The straightforward enantioselective construction of the hydroquinoline ring system from 1,5-polycarbonyl derivatives, using (R)-phenyglycinol as a chiral latent form of ammonia, is reported. The process mimics the key steps believed to occur in nature in the biosynthesis of amphibian decahydroquinoline alkaloids. Diastereodivergent routes to enantiopure cis-2,5-disubstituted decahydroquinolines, including the alkaloid pumiliotoxin C (cis-195A), are developed.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Biomimetics / methods*
  • Molecular Mimicry
  • Quinolines / chemical synthesis*
  • Stereoisomerism

Substances

  • Quinolines