Regulation of glutathione S-transferase gene expression by phenobarbital in cultured adult rat hepatocytes

FEBS Lett. 1991 Jun 17;284(1):103-8. doi: 10.1016/0014-5793(91)80772-u.

Abstract

Previous studies, by using Northern blotting analyses, showed that phenobarbital (PB) affects the steady-state mRNA levels of glutathione S-transferase (GST) subunits 1/2, 3/4 and 7 in both conventional cultures of adult rat hepatocytes and co-cultures, with rat liver epithelial cells [Vandenberghe et al., 1989, FEBS Lett. 251, 59-64; Morel et al., 1989, FEBS Lett. 258, 99-102]. To determine whether PB acts at the transcriptional level, nuclear 'run on' experiments using cDNA probes hybridizing to GST subunits 1/2, 3/4 and 7 mRNA were performed on purified nuclei isolated from control and PB treated hepatocytes seeded under conventional and co-culture conditions. Data from this study demonstrate that the increase in steady-state mRNA levels observed in both conventional culture and co-culture after 4 days PB exposure results from an increased transcriptional activity of the GST genes. However, a substantial increase in steady-state mRNA levels in the absence of a commensurate increase in transcriptional activity at 12 days of co-culture, indicates that the barbiturate has also a stabilizing effect in vitro on the GST mRNAs.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cells, Cultured
  • Gene Expression Regulation, Enzymologic / drug effects*
  • Glutathione Transferase / genetics*
  • Glutathione Transferase / metabolism
  • Liver / cytology
  • Liver / enzymology*
  • Phenobarbital / pharmacology*
  • Rats
  • Rats, Inbred Strains
  • Transcription, Genetic

Substances

  • Glutathione Transferase
  • Phenobarbital