Atorvastatin has antithrombotic effects in patients with type 1 diabetes and dyslipidemia

Thromb Res. 2010 Sep;126(3):e225-31. doi: 10.1016/j.thromres.2010.05.023. Epub 2010 Jul 15.

Abstract

Introduction: Diabetes is a prothrombotic state involving a more thrombogenic fibrin network. In the present study we investigated the effects of lipid-lowering therapy with atorvastatin on fibrin network structure and platelet-derived microparticles in patients with type 1 diabetes and dyslipidemia.

Materials and methods: Twenty patients were treated with atorvastatin (80 mg daily) or placebo during 2 months in a randomized, double-blind, cross-over study. Fibrin network permeability, expression of glycoprotein IIIa, P-selectin and tissue factor on platelet-derived microparticles, plasma endogenous thrombin potential, plasminogen activator inhibitor-1 and tissue plasminogen activator antigen levels were assessed. Additionally, levels of plasma fibrinogen, high-sensitivity C-reactive protein and glycated haemoglobin were measured.

Results: During treatment with atorvastatin, fibrin network permeability increased (p=0.01), while endogenous thrombin potential and expression of glycoprotein IIIa, P-selectin and tissue factor decreased (p<0.01). In vitro experiments indicated that platelet-derived microparticles influence the fibrin network formation as fibrin network permeability decreased significantly when platelet-derived microparticles were added to normal plasma. Baseline levels of plasminogen activator inhibitor-1 and tissue plasminogen activator antigen as well as plasma fibrinogen and high-sensitivity C-reactive protein were within reference values and not significantly changed during atorvastatin treatment, while glycated haemoglobin increased 0.3% (p<0.001).

Conclusions: Novel treatment effects were found in patients with type 1 diabetes and dyslipidemia during atorvastatin therapy, i.e. a more porous fibrin network, to which reduced expression of glycoprotein IIIa, P-selectin and tissue factor on platelet-derived microparticles may contribute. The observed impairment of glycemic control during long-term statin treatment deserves attention.

Publication types

  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Aged
  • Atorvastatin
  • Biomarkers / blood
  • Blood Platelets / drug effects
  • Blood Platelets / metabolism
  • C-Reactive Protein / metabolism
  • Cell-Derived Microparticles / drug effects
  • Cell-Derived Microparticles / metabolism
  • Cross-Over Studies
  • Diabetes Mellitus, Type 1 / blood
  • Diabetes Mellitus, Type 1 / complications*
  • Double-Blind Method
  • Dyslipidemias / blood
  • Dyslipidemias / complications
  • Dyslipidemias / drug therapy*
  • Fibrin / metabolism
  • Fibrinolytic Agents / therapeutic use*
  • Glycated Hemoglobin / metabolism
  • Heptanoic Acids / therapeutic use*
  • Humans
  • Hydroxymethylglutaryl-CoA Reductase Inhibitors / therapeutic use*
  • Integrin beta3 / blood
  • Middle Aged
  • P-Selectin / blood
  • Plasminogen Activator Inhibitor 1 / blood
  • Pyrroles / therapeutic use*
  • Sweden
  • Thrombin / metabolism
  • Thromboplastin / metabolism
  • Thrombosis / blood
  • Thrombosis / drug therapy*
  • Thrombosis / etiology
  • Time Factors
  • Treatment Outcome

Substances

  • Biomarkers
  • Fibrinolytic Agents
  • Glycated Hemoglobin A
  • Heptanoic Acids
  • Hydroxymethylglutaryl-CoA Reductase Inhibitors
  • Integrin beta3
  • P-Selectin
  • Plasminogen Activator Inhibitor 1
  • Pyrroles
  • SERPINE1 protein, human
  • hemoglobin A1c protein, human
  • Fibrin
  • C-Reactive Protein
  • Thromboplastin
  • Atorvastatin
  • Thrombin