[Effects of Ginkgolide B on inflammation induced by cerebral ischemia-reperfusion in rats]

Zhong Yao Cai. 2010 Apr;33(4):578-80.
[Article in Chinese]

Abstract

Objective: To investigate the protective effects of Ginkgolide B on inflammation induced by cerebral ischemia-reperfusion in rats.

Methods: Rats were pretreated with Ginkgolide B at the dose of 2. 5, 5, 10 mg/kg for 3 days and then subjected to cerebral ischemia/reperfusion induced by a middle cerebral artery occlusion (MCAO). The infarct volume and the neurological deficit were determined by the method of TTC (2,3,5-triphenylterazolium chloride) staining and Longa's score. The permeability of blood-brain barrier (BBB) was evaluated by measurement of the evans blue (EB) content in the brain with spectrophotometer. The content of interleukin-1beta, interleukin-6 (IL-6, IL-1beta) in serum and tumor necrosis factor-alpha (TNF-alpha), The content of E-selectin and ICAM 1 in brain were determined by radio-immunoassay and ELISA assay.

Results: Ginkgolide B reduced infarct volume, ameliorated the neurological deficit and the permeability of BBB, the content of IL-6, IL-1beta in serum and TNF-alpha, expressions of E-selectin and ICAM 1 in brain tissue also were significantly decreased.

Conclusion: Ginkgolide B has protective effects on cerebral injury by inhibiting the inflammation induced by ischemia/reperfusion injury.

MeSH terms

  • Animals
  • Blood-Brain Barrier / drug effects
  • Blood-Brain Barrier / pathology
  • Brain / drug effects
  • Brain / metabolism
  • Brain / pathology
  • Brain Ischemia / complications*
  • Disease Models, Animal
  • E-Selectin / metabolism
  • Ginkgo biloba / chemistry*
  • Ginkgolides / administration & dosage
  • Ginkgolides / pharmacology*
  • Infarction, Middle Cerebral Artery / blood
  • Infarction, Middle Cerebral Artery / etiology
  • Infarction, Middle Cerebral Artery / prevention & control*
  • Inflammation Mediators / blood*
  • Inflammation Mediators / metabolism
  • Interleukin-1beta / blood
  • Interleukin-6 / blood
  • Lactones / administration & dosage
  • Lactones / pharmacology*
  • Male
  • Neuroprotective Agents / pharmacology
  • Plant Leaves / chemistry
  • Random Allocation
  • Rats
  • Rats, Sprague-Dawley
  • Reperfusion Injury / complications*
  • Tumor Necrosis Factor-alpha / metabolism

Substances

  • E-Selectin
  • Ginkgolides
  • Inflammation Mediators
  • Interleukin-1beta
  • Interleukin-6
  • Lactones
  • Neuroprotective Agents
  • Tumor Necrosis Factor-alpha
  • ginkgolide B