Benefit of magnesium-25 carrying porphyrin-fullerene nanoparticles in experimental diabetic neuropathy

Int J Nanomedicine. 2010 Aug 9:5:517-23. doi: 10.2147/ijn.s11643.

Abstract

Diabetic neuropathy (DN) is a debilitating disorder occurring in most diabetic patients without a viable treatment yet. The present work examined the protective effect of (25)Mg-PMC(16) nanoparticle (porphyrin adducts of cyclohexil fullerene-C60) in a rat model of streptozotocin (STZ)-induced DN. (25)Mg-PMC(16) (0.5 lethal dose(50) [LD(50)]) was administered intravenously in two consecutive days before intraperitoneal injection of STZ (45 mg/kg). (24)Mg-PMC(16) and MgCl(2) were used as controls. Blood 2,3-diphosphoglycerate (2,3-DPG), oxidative stress biomarkers, adenosine triphosphate (ATP) level in dorsal root ganglion (DRG) neurons were determined as biomarkers of DN. Results indicated that 2,3-DPG and ATP decreased whereas oxidative stress increased by induction of DN which all were improved in (25)Mg-PMC(16)-treated animals. No significant changes were observed by administration of (24)Mg-PMC(16) or MgCl(2) in DN rats. It is concluded that in DN, oxidative stress initiates injuries to DRG neurons that finally results in death of neurons whereas administration of (25)Mg-PMC(16) by release of Mg and increasing ATP acts protectively.

Keywords: 25Mg-magnetic isotope effect; adenosine triphosphate; diabetes; nanotechnology; neuropathy; oxidative stress; porphyrin-fullerene nanoparticles.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 2,3-Diphosphoglycerate / blood
  • Adenosine Diphosphate / metabolism
  • Adenosine Triphosphate / metabolism
  • Animals
  • Diabetic Neuropathies / drug therapy*
  • Diabetic Neuropathies / metabolism
  • Diabetic Neuropathies / pathology
  • Drug Delivery Systems
  • Fullerenes / chemistry
  • Ganglia, Spinal / drug effects
  • Ganglia, Spinal / metabolism
  • Humans
  • Isotopes / administration & dosage
  • Magnesium / administration & dosage*
  • Magnesium / metabolism
  • Male
  • Nanomedicine
  • Nanoparticles / administration & dosage*
  • Nanoparticles / chemistry*
  • Oxidative Stress / drug effects
  • Porphyrins / chemistry
  • Rats
  • Rats, Wistar

Substances

  • Fullerenes
  • Isotopes
  • Porphyrins
  • 2,3-Diphosphoglycerate
  • Adenosine Diphosphate
  • Adenosine Triphosphate
  • Magnesium
  • fullerene C60