[Causes of selectivity, activation and inhibition. Molecular mechanisms of endothelin-receptor recognition]

Pharm Unserer Zeit. 2010 Nov;39(6):442-7. doi: 10.1002/pauz.201000389.
[Article in German]
No abstract available

Publication types

  • Review

MeSH terms

  • Amino Acid Sequence
  • Antihypertensive Agents / metabolism
  • Antihypertensive Agents / pharmacology
  • Bosentan
  • Endothelin Receptor Antagonists*
  • Humans
  • Isoxazoles / metabolism
  • Isoxazoles / pharmacology
  • Ligands
  • Models, Molecular
  • Molecular Sequence Data
  • Receptors, Endothelin / drug effects
  • Receptors, Endothelin / genetics*
  • Sulfonamides / metabolism
  • Sulfonamides / pharmacology
  • Thiophenes / metabolism
  • Thiophenes / pharmacology

Substances

  • Antihypertensive Agents
  • Endothelin Receptor Antagonists
  • Isoxazoles
  • Ligands
  • Receptors, Endothelin
  • Sulfonamides
  • Thiophenes
  • sitaxsentan
  • Bosentan