Calcineurin inhibitors in pediatric atopic dermatitis: a review of current evidence

Am J Clin Dermatol. 2011 Feb 1;12(1):15-24. doi: 10.2165/11319300-000000000-00000.

Abstract

Atopic dermatitis (AD) is a common, chronic inflammatory dermatosis with a prevalence of 7-21% in school-aged children. Childhood AD has a profound impact on the social, personal, emotional, and financial perspectives of families. For the last half-century, topical corticosteroids of different potencies have been the mainstay of topical therapy. In recent years, two topical calcineurin inhibitors (TCIs), tacrolimus and pimecrolimus, have become available for the treatment of AD. Both tacrolimus and pimecrolimus have been extensively evaluated in the management of pediatric AD. Trials comparing them with placebo, topical corticosteroids, and each other have shown them to be effective and safe for continuous short-term use, and for noncontinuous use for up to 4 years. Long-term safety of TCIs is not known as they have been in clinical use for less than a decade.

Publication types

  • Comparative Study
  • Review

MeSH terms

  • Administration, Cutaneous
  • Animals
  • Calcineurin Inhibitors*
  • Child
  • Dermatitis, Atopic / drug therapy*
  • Dermatitis, Atopic / physiopathology
  • Dermatologic Agents / adverse effects
  • Dermatologic Agents / pharmacology
  • Dermatologic Agents / therapeutic use*
  • Glucocorticoids / adverse effects
  • Glucocorticoids / therapeutic use
  • Humans
  • Immunosuppressive Agents / adverse effects
  • Immunosuppressive Agents / pharmacology
  • Immunosuppressive Agents / therapeutic use
  • Tacrolimus / adverse effects
  • Tacrolimus / analogs & derivatives*
  • Tacrolimus / pharmacology
  • Tacrolimus / therapeutic use

Substances

  • Calcineurin Inhibitors
  • Dermatologic Agents
  • Glucocorticoids
  • Immunosuppressive Agents
  • pimecrolimus
  • Tacrolimus