High-fat feeding promotes obesity via insulin receptor/PI3K-dependent inhibition of SF-1 VMH neurons

Nat Neurosci. 2011 Jun 5;14(7):911-8. doi: 10.1038/nn.2847.

Abstract

Steroidogenic factor 1 (SF-1)-expressing neurons of the ventromedial hypothalamus (VMH) control energy homeostasis, but the role of insulin action in these cells remains undefined. We show that insulin activates phosphatidylinositol-3-OH kinase (PI3K) signaling in SF-1 neurons and reduces firing frequency in these cells through activation of K(ATP) channels. These effects were abrogated in mice with insulin receptor deficiency restricted to SF-1 neurons (SF-1(ΔIR) mice). Whereas body weight and glucose homeostasis remained the same in SF-1(ΔIR) mice as in controls under a normal chow diet, they were protected from diet-induced leptin resistance, weight gain, adiposity and impaired glucose tolerance. High-fat feeding activated PI3K signaling in SF-1 neurons of control mice, and this response was attenuated in the VMH of SF-1(ΔIR) mice. Mimicking diet-induced overactivation of PI3K signaling by disruption of the phosphatidylinositol-3,4,5-trisphosphate phosphatase PTEN led to increased body weight and hyperphagia under a normal chow diet. Collectively, our experiments reveal that high-fat diet-induced, insulin-dependent PI3K activation in VMH neurons contributes to obesity development.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Action Potentials / drug effects
  • Action Potentials / genetics
  • Age Factors
  • Animals
  • Animals, Newborn
  • Blood Glucose / drug effects
  • Body Weight / drug effects
  • Calorimetry / methods
  • Dietary Fats / adverse effects*
  • Dose-Response Relationship, Drug
  • Eating / drug effects
  • Eating / physiology
  • Enzyme Inhibitors / pharmacology
  • Enzyme-Linked Immunosorbent Assay / methods
  • Female
  • Gene Expression Regulation / drug effects
  • Glucose Tolerance Test
  • Green Fluorescent Proteins / genetics
  • Hypoglycemic Agents / pharmacology
  • In Vitro Techniques
  • Injections, Intraventricular / methods
  • Insulin / pharmacology
  • Leptin / administration & dosage
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Mice, Transgenic
  • Neurons / drug effects*
  • Neurons / metabolism
  • Obesity / chemically induced*
  • Obesity / pathology*
  • Patch-Clamp Techniques
  • Phosphatidylinositol 3-Kinases / metabolism*
  • RNA, Messenger / metabolism
  • Receptor, Insulin / metabolism*
  • Signal Transduction / drug effects
  • Signal Transduction / genetics
  • Steroidogenic Factor 1 / genetics
  • Steroidogenic Factor 1 / metabolism
  • Time Factors
  • Tolbutamide / pharmacology
  • Ventromedial Hypothalamic Nucleus / cytology
  • Ventromedial Hypothalamic Nucleus / pathology*

Substances

  • Blood Glucose
  • Dietary Fats
  • Enzyme Inhibitors
  • Hypoglycemic Agents
  • Insulin
  • Leptin
  • RNA, Messenger
  • Steroidogenic Factor 1
  • steroidogenic factor 1, mouse
  • Green Fluorescent Proteins
  • Tolbutamide
  • Phosphatidylinositol 3-Kinases
  • Receptor, Insulin