Irsogladine maleate regulates epithelial barrier function in tumor necrosis factor-α-stimulated human gingival epithelial cells

J Periodontal Res. 2012 Feb;47(1):55-61. doi: 10.1111/j.1600-0765.2011.01404.x. Epub 2011 Sep 6.

Abstract

Background and objective: As epithelial cells function as a mechanical barrier, the permeability of the gingival epithelial cell layer indicates a defensive capability against invasion by periodontal pathogens. We have reported the expression of claudin-1 and E-cadherin, key regulators of permeability, in the gingival junctional epithelium. Irsogladine maleate (IM) is a medication for gastric ulcers and also regulates Aggregatibacter actinomycetemcomitans-stimuated chemokine secretion and E-cadherin expression in gingival epithelium. In this study, we have further investigated the effects of IM on the barrier functions of gingival epithelial cells under inflammatory conditions.

Material and methods: We examined the permeability, and the expression of claudin-1 and E-cadherin, in human gingival epithelial cells (HGECs) stimulated with tumor necrosis factor (TNF)-α, with or without IM.

Results: TNF-α increased the permeability of HGECs, and IM abolished the increase. TNF-α reduced the expression of E-cadherin in HGECs, and IM reversed the reduction. In addition, immunofluorescence staining showed that TNF-α disrupted claudin-1 expression in HGECs, and IM reversed this effect.

Conclusion: The results suggest that IM reverses the TNF-α-induced disruption of the gingival epithelial barrier by regulating E-cadherin and claudin-1.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Blotting, Western
  • Cadherins / drug effects
  • Cell Culture Techniques
  • Cell Line
  • Cell Membrane Permeability / drug effects
  • Claudin-1
  • Electric Impedance
  • Epithelial Attachment / cytology
  • Epithelial Attachment / drug effects
  • Epithelial Cells / drug effects
  • Epithelial Cells / immunology
  • Female
  • Fluorescein
  • Fluorescent Antibody Technique
  • Fluorescent Dyes
  • Gingiva / cytology
  • Gingiva / drug effects*
  • Gingiva / immunology
  • Humans
  • Male
  • Membrane Proteins / drug effects
  • Real-Time Polymerase Chain Reaction
  • Tight Junctions / drug effects
  • Triazines / pharmacology*
  • Tumor Necrosis Factor-alpha / antagonists & inhibitors
  • Tumor Necrosis Factor-alpha / pharmacology*
  • Young Adult

Substances

  • CLDN1 protein, human
  • Cadherins
  • Claudin-1
  • Fluorescent Dyes
  • Membrane Proteins
  • Triazines
  • Tumor Necrosis Factor-alpha
  • irsogladine
  • Fluorescein