Renal effects of long-term darbepoetin alpha treatment in hypertensive TGR(mRen2)27 rats

J Renin Angiotensin Aldosterone Syst. 2012 Jun;13(2):232-8. doi: 10.1177/1470320311432186. Epub 2012 Jan 26.

Abstract

Introduction: Erytropoietin (EPO) has cytoprotective and angiogenic properties and has a beneficial effect in ischaemic conditions. Since the development of renal interstitial abnormalities are often associated with ischaemia, we studied the effects of the long-acting EPO analogue darbepoetin alpha (DA) on kidney damage in TGR(mRen2)27 (Ren2) rats.

Materials and methods: Ren2 rats were randomised to DA or vehicle (VEH) or to DA + angiotensin converting enzyme inhibitor (ACEi) or VEH + ACEi. Sprague Dawley (SD) rats served as controls. Blood pressure was measured weekly and 24-h urine was collected to measure proteinuria. Blood samples were collected for creatinine and haematocrit. Kidneys were studied for inflammation and pre-fibrosis. Renal mRNA expression was studied for EPO, EPO-receptor, collagen-3α1 and kidney injury molecule-1 (KIM-1).

Results: DA had no effect on SBP, serum creatinine and proteinuria. Interstitial and glomerular α-SMA expression was significantly increased in Ren2. ACEi but not DA improved the increased renal inflammatory and pro-fibrotic profile in Ren2 rats. DA on top of ACEi further reduced glomerular α-SMA and KIM-1 expression.

Conclusion: Long-term DA treatment has no beneficial effects on renal structural and functional changes in TGR(mRen2)27 rats in the time frame studied and the dose provided.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Actins / metabolism
  • Animals
  • Cell Adhesion Molecules / genetics
  • Cell Adhesion Molecules / metabolism
  • Cell Count
  • Collagen Type III / genetics
  • Collagen Type III / metabolism
  • Darbepoetin alfa
  • Disease Models, Animal
  • Erythropoietin / analogs & derivatives*
  • Erythropoietin / pharmacology
  • Gene Expression Regulation / drug effects
  • Hypertension / pathology
  • Hypertension / physiopathology*
  • Kidney / drug effects*
  • Kidney / pathology*
  • Kidney / physiopathology
  • Kidney Glomerulus / drug effects
  • Kidney Glomerulus / pathology
  • Kidney Glomerulus / physiopathology
  • Macrophages / drug effects
  • Macrophages / pathology
  • Male
  • RNA, Messenger / genetics
  • RNA, Messenger / metabolism
  • Rats
  • Receptors, Erythropoietin / genetics
  • Receptors, Erythropoietin / metabolism
  • Time Factors

Substances

  • Actins
  • Cell Adhesion Molecules
  • Collagen Type III
  • Havcr1protein, rat
  • RNA, Messenger
  • Receptors, Erythropoietin
  • smooth muscle actin, rat
  • Erythropoietin
  • Darbepoetin alfa