Ascorbate antagonizes nickel ion to regulate JMJD1A expression in kidney cancer cells

Acta Biochim Biophys Sin (Shanghai). 2012 Apr;44(4):330-8. doi: 10.1093/abbs/gms004. Epub 2012 Feb 7.

Abstract

Abnormal expression of histone demethylase Jumonji domain-containing protein 1A (JMJD1A) is associated with many kinds of cancers. JMJD1A is also a hypoxic response gene and its expression is regulated by hypoxia-inducible factor-1α (HIF-1α). In this study, we determined the role of JMJD1A in development and hypoxia pathway. We also measured the expression of JMJD1A and two hypoxia factors glucose transporter 1 (GLUT1) and vascular endothelial growth factor (VEGF) in 786-0 and HEK293 cells treated with different concentrations of NiCl(2) (2.5-100 μM) for 24 h, and found that JMJD1A mRNA and protein were up-regulated with increased concentrations of NiCl(2). We then observed that ascorbate could retard the up-regulated effect of NiCl(2)-induced JMJD1A expression in a dose-dependent manner through decreasing the stability of HIF-1α protein. Immunohistochemical analysis further demonstrated ascorbate antagonized Ni(2+)-induced up-regulation of JMJD1A expression in 786-0, HEK293, and OS-RC-2 cells. These findings suggest that both Ni(2+) and ascorbate can regulate the expression of histone demethylase JMJD1A, which is important for cancer development or inhibition.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antioxidants / pharmacology
  • Ascorbic Acid / pharmacology*
  • Blotting, Western
  • Cell Line, Tumor
  • Dose-Response Relationship, Drug
  • Drug Antagonism
  • Gene Expression Regulation, Neoplastic / drug effects*
  • HEK293 Cells
  • Humans
  • Hypoxia-Inducible Factor 1, alpha Subunit / metabolism
  • Immunohistochemistry
  • Jumonji Domain-Containing Histone Demethylases / genetics*
  • Jumonji Domain-Containing Histone Demethylases / metabolism
  • Kidney / drug effects
  • Kidney / metabolism
  • Kidney Neoplasms / genetics
  • Kidney Neoplasms / metabolism
  • Kidney Neoplasms / pathology
  • Male
  • Mice
  • Mice, Inbred BALB C
  • Nickel / pharmacology*
  • Reverse Transcriptase Polymerase Chain Reaction

Substances

  • Antioxidants
  • Hypoxia-Inducible Factor 1, alpha Subunit
  • nickel chloride
  • Nickel
  • Jumonji Domain-Containing Histone Demethylases
  • KDM3A protein, human
  • Ascorbic Acid