Effects of N1-methylnicotinamide on oxidative and glycooxidative stress markers in rats with streptozotocin-induced diabetes mellitus

Redox Rep. 2012;17(1):1-7. doi: 10.1179/1351000211Y.0000000016.

Abstract

Objectives: This study was focused on the monitoring how the anti-inflammatory substance, N(1)-methylnicotinamide (MNA), could influence oxidation and glycooxidation stress markers in rats under conditions of streptozotocin (STZ)-induced diabetes mellitus.

Methods: Diabetes mellitus was induced in 60 male Wistar rats by intraperitoneal injection of STZ and after 7 days diabetic animals were allocated to five groups according to the dose of MNA administered for 7 weeks. The degree of DNA damage in lymphocytes, as well as advanced glycation endproducts (AGEs), protein carbonyls, lipid peroxides, and total antioxidant capacity (TEAC) in plasma were measured.

Results: Glycation damage to proteins (represented by AGEs level) was significantly increased in all diabetic groups compared to untreated non-diabetic animals. MNA did not affect TEAC of plasma in any group of diabetic rats. Supplementation of diabetic rats with MNA at the dose of 200 mg/kg resulted in decreased protein carbonyls (from 0.0818±0.0091 to 0.0558±0.0044 nmol/mg proteins; P<0.05, n=15) and DNA oxidation, reflected by the levels of 8-oxoG (0.6302±0.085 vs. 0.9213±0.108 8-oxoG/10(6) G; P<0.05, n=15), compared to untreated diabetic animals.

Discussion: Our results demonstrated that MNA at suitable concentrations could influence oxidative modifications of proteins and DNA.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antioxidants / metabolism
  • Biomarkers / analysis
  • DNA Damage
  • Diabetes Mellitus, Experimental / metabolism*
  • Diabetes Mellitus, Experimental / pathology
  • Drug Evaluation, Preclinical
  • Glycation End Products, Advanced / analysis
  • Lipid Peroxidation / drug effects
  • Lipid Peroxides / blood
  • Lymphocytes / metabolism
  • Lymphocytes / pathology
  • Male
  • Niacinamide / analogs & derivatives*
  • Niacinamide / pharmacology
  • Oxidation-Reduction
  • Oxidative Stress*
  • Protein Carbonylation / drug effects
  • Rats
  • Rats, Wistar
  • Streptozocin

Substances

  • Antioxidants
  • Biomarkers
  • Glycation End Products, Advanced
  • Lipid Peroxides
  • Niacinamide
  • Streptozocin
  • N(1)-methylnicotinamide