Effects of corneal thickness on the intraocular penetration of travoprost 0.004%

Eye (Lond). 2012 Jul;26(7):972-5. doi: 10.1038/eye.2012.74. Epub 2012 May 4.

Abstract

Purpose: To determine whether the intraocular penetration of travoprost 0.004% is affected by central corneal thickness.

Methods: Sixty-four patients who were scheduled for cataract surgery without any other ophthalmologic pathology of significance were enrolled in this study. At 120 min before surgery, one drop of travoprost 0.004% was instilled in the eye to be operated on. At the start of surgery, a sample of aqueous humour was extracted to subsequently determine its AL-5848 concentration. These concentrations were compared among three groups of patients established according to central corneal thickness measurements obtained by ultrasound pachymetry.

Results: Mean AL-5848 concentrations were 3.27±2.03 ng/ml in Group I (CCT<511 microns), 3.27±2.44 ng/ml in Group II (CCT≥511 and ≤574 microns), and 2.73±2.15 ng/ml in Group III (CCT>574 microns), indicating no significant differences among the groups.

Conclusions: We were unable to demonstrate the greater or lesser penetration of travoprost depending on corneal thickness, which could explain differences in patient responses to this drug.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Antihypertensive Agents / pharmacokinetics*
  • Antihypertensive Agents / therapeutic use
  • Aqueous Humor / metabolism*
  • Cloprostenol / analogs & derivatives*
  • Cloprostenol / pharmacokinetics
  • Cloprostenol / therapeutic use
  • Cornea / anatomy & histology*
  • Cornea / metabolism
  • Female
  • Glaucoma / drug therapy
  • Glaucoma / metabolism*
  • Humans
  • Male
  • Travoprost

Substances

  • Antihypertensive Agents
  • Cloprostenol
  • Travoprost