Effects of hydroquinone on retinal and vascular cells in vitro

Indian J Ophthalmol. 2012 May-Jun;60(3):189-93. doi: 10.4103/0301-4738.95869.

Abstract

Aim: To explore the molecular pathophysiology that might explain the epidemiologic association between cigarette smoke and age-related macular degeneration (AMD) by examining the effects of hydroquinone (HQ), a toxic compound present in high concentration in cigarette smoke-related tar, on human retinal pigment epithelial cells (ARPE-19), rat retinal neurosensory cells (R-28), and human microvascular endothelial cells (HMVEC).

Materials and methods: ARPE-19, R-28, and HMVEC were treated for 24 h with four different concentrations of HQ (500 μM, 200 μM, 100 μM, 50 μM). Cell viability, caspase-3/7 activation, DNA laddering patterns, and lactate dehydrogenase (LDH) levels were analyzed.

Results: At 50 μM HQ, R-28 cells showed a significant decrease in cell viability compared with the dimethyl sulfoxide (DMSO)-treated controls. At the 100-500 μM concentrations, all three cell lines showed significant cell death (P < 0.001). In the ARPE-19, R-28, and HMVEC cultures, the caspase-3/7 activities were not increased at any of the HQ concentration.

Conclusion: Our findings suggest that the mechanism of cell death in all three cell lines was through non-apoptotic pathway. In addition, neuroretinal R-28 cells were more sensitive to HQ than the ARPE-19 and HMVEC cultures.

Publication types

  • Comparative Study

MeSH terms

  • Animals
  • Animals, Newborn
  • Apoptosis / drug effects
  • Caspase 3 / metabolism
  • Caspase 7 / metabolism
  • Cell Survival
  • Cells, Cultured
  • DNA Fragmentation / drug effects
  • Disease Models, Animal
  • Endothelium, Vascular / drug effects*
  • Endothelium, Vascular / enzymology
  • Endothelium, Vascular / pathology
  • Humans
  • Hydroquinones / toxicity*
  • Macular Degeneration / chemically induced
  • Macular Degeneration / genetics
  • Macular Degeneration / pathology*
  • Mutagens / toxicity
  • Rats
  • Retinal Pigment Epithelium / drug effects*
  • Retinal Pigment Epithelium / enzymology
  • Retinal Pigment Epithelium / pathology

Substances

  • Hydroquinones
  • Mutagens
  • Caspase 3
  • Caspase 7
  • hydroquinone