Trimetazidine and inflammatory response in coronary artery bypass grafting

Arq Bras Cardiol. 2012 Aug;99(2):688-96. doi: 10.1590/s0066-782x2012005000066. Epub 2012 Jul 13.
[Article in English, Portuguese]

Abstract

Background: Organic inflammatory response is a pathophysiological mechanism present at every coronary artery bypass grafting with extracorporeal circulation (CABG-ECC), the release of inflammatory mediators being one of its defense mechanisms.

Objective: To assess, in a prospective double-blind randomized and placebo-controlled study, the effects of trimetazidine (Tmz) on the inflammatory response, by using the variation in interleukins 6 and 8, TNF-α, complements C3 and C5, and highly sensitive C-reactive protein (HS-CRP) levels in the pre- and post-operative periods.

Methods: This study assessed 30 patients undergoing CABG-ECC with intermittent hypothermic cardioplegia, and having, at most, mild ventricular dysfunction. The patients were divided into two groups (placebo and Tmz), stratified by echocardiography, and received drug/placebo at the dose of 60 mg/day. Measurements were taken as follows: in the pre-operative period with no drug; on the day of surgery, corresponding to 12 to 15 days on drug/placebo; five minutes after aortic unclamping; 12 and 24 hours after surgery, for interleukins and complements; and 48 hours after surgery, for HS-CRP.

Results: No significant difference between the levels of interleukin 8, TNF-α, C3 and C5, and HS-CRP was observed. However, the interleukin 6 levels were significantly lower in the group treated as compared with those in the control group at all time points assessed.

Conclusion: Trimetazidine proved to be effective only for reducing interleukin 6 in patients undergoing CABG.

Publication types

  • Randomized Controlled Trial

MeSH terms

  • Aged
  • Biomarkers / blood
  • Coronary Artery Bypass / methods*
  • Cytokines / blood
  • Double-Blind Method
  • Female
  • Humans
  • Inflammation / metabolism
  • Inflammation Mediators / metabolism
  • Male
  • Placebos / administration & dosage
  • Postoperative Period
  • Prospective Studies
  • Time Factors
  • Treatment Outcome
  • Trimetazidine / administration & dosage*
  • Vasodilator Agents / administration & dosage*

Substances

  • Biomarkers
  • Cytokines
  • Inflammation Mediators
  • Placebos
  • Vasodilator Agents
  • Trimetazidine