Evidence that the 5-HT1A receptor agonists buspirone and ipsapirone activate adrenaline release in the conscious rat

Eur J Pharmacol. 1990 Feb 20;177(1-2):107-10. doi: 10.1016/0014-2999(90)90558-n.

Abstract

The aim of this study was to investigate the effects of the 5-HT1A receptor agonists buspirone and ipsapirone (1-10 mg/kg) on plasma adrenaline (A) levels and on glycemia in the conscious rat. The results indicate that buspirone was able, within 5 min, to increase plasma A and glucose levels in a dose-dependent manner. Ipsapirone administration triggered similar patterns, except that the highest dose used (10 mg/kg) promoted a time-dependent increase in plasma A and glucose levels that was maximal at the end of analysis.

MeSH terms

  • Animals
  • Blood Glucose / metabolism
  • Buspirone / pharmacology*
  • Chromatography, High Pressure Liquid
  • Dose-Response Relationship, Drug
  • Epinephrine / blood
  • Epinephrine / metabolism*
  • Male
  • Pyrimidines / pharmacology*
  • Rats
  • Rats, Inbred Strains
  • Receptors, Serotonin / drug effects
  • Receptors, Serotonin / metabolism*

Substances

  • Blood Glucose
  • Pyrimidines
  • Receptors, Serotonin
  • ipsapirone
  • Buspirone
  • Epinephrine