Npas4 is a novel activity-regulated cytoprotective factor in pancreatic β-cells

Diabetes. 2013 Aug;62(8):2808-20. doi: 10.2337/db12-1527. Epub 2013 May 8.

Abstract

Cellular homeostasis requires intrinsic sensing mechanisms to temper function in the face of prolonged activity. In the pancreatic β-cell, glucose is likely a physiological trigger that activates an adaptive response to stimulation, thereby maintaining cellular homeostasis. Immediate early genes (IEGs) are activated as a first line of defense in cellular homeostasis and are largely responsible for transmitting an environmental cue to a cellular response. Here we examine the regulation and function of the novel β-cell IEG, neuronal PAS domain protein 4 (Npas4). Using MIN6 cells, mouse and human islets, as well as in vivo infusions, we demonstrate that Npas4 is expressed within pancreatic islets and is upregulated by β-cell depolarizing agents. Npas4 tempers β-cell function through a direct inhibitory interaction with the insulin promoter and by blocking the potentiating effects of GLP-1 without significantly reducing glucose-stimulated secretion. Finally, Npas4 expression is induced by classical endoplasmic reticulum (ER) stressors and can prevent thapsigargin- and palmitate-induced dysfunction and cell death. These results suggest that Npas4 is a key activity-dependent regulator that improves β-cell efficiency in the face of stress. We posit that Npas4 could be a novel therapeutic target in type 2 diabetes that could both reduce ER stress and cell death and maintain basal cell function.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Basic Helix-Loop-Helix Transcription Factors / genetics
  • Basic Helix-Loop-Helix Transcription Factors / metabolism*
  • Cell Line
  • Cytoprotection / drug effects
  • Cytoprotection / genetics*
  • Emulsions / pharmacology
  • Endoplasmic Reticulum Stress / physiology
  • Glucagon-Like Peptide 1 / pharmacology
  • Glucose / pharmacology
  • Humans
  • Insulin / genetics
  • Insulin / metabolism
  • Insulin-Secreting Cells / drug effects
  • Insulin-Secreting Cells / metabolism*
  • Islets of Langerhans / drug effects
  • Islets of Langerhans / metabolism*
  • Mice
  • Phospholipids / pharmacology
  • Promoter Regions, Genetic
  • Soybean Oil / pharmacology
  • Up-Regulation / drug effects

Substances

  • Basic Helix-Loop-Helix Transcription Factors
  • Emulsions
  • Insulin
  • Npas4 protein, mouse
  • Phospholipids
  • soybean oil, phospholipid emulsion
  • Soybean Oil
  • Glucagon-Like Peptide 1
  • Glucose