Anti-platelet therapy in the prevention of hepatitis B virus-associated hepatocellular carcinoma

J Hepatol. 2013 Nov;59(5):1135-8. doi: 10.1016/j.jhep.2013.05.040. Epub 2013 Jun 4.

Abstract

Previous studies in mouse models of self-limited viral hepatitis showed that platelets contribute to acute liver damage by promoting the intrahepatic accumulation of virus-specific CD8 T cells and, secondarily, virus-non-specific inflammatory cells. Built on these observations, a recent preclinical study took advantage of a previously established hepatitis B virus (HBV) transgenic mouse model of immune-mediated chronic hepatitis that progresses to hepatocellular carcinoma (HCC), to demonstrate that clinically achievable doses of the anti-platelet drugs aspirin and clopidogrel - administered continuously after the onset of liver disease - can prevent hepatocarcinogenesis and greatly improve overall survival. These outcomes were preceded by and associated with reduced hepatic accumulation of virus-specific CD8 T cells and virus-non-specific inflammatory cells, reduced hepatocellular injury and hepatocellular proliferation, and reduced severity of liver fibrosis. The observation that anti-platelet therapy inhibits HCC development identifies platelets as key players in the pathogenesis of HBV-associated liver cancer and supports the notion that a sustained immune-mediated necroinflammatory liver disease is sufficient to trigger HCC. The results abovementioned and their clinical implications are discussed in this report.

Keywords: Anti-platelet drugs; CD8 T cells; Hepatitis B virus; Hepatocellular carcinoma; Platelets; Viral hepatitis.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Aspirin / pharmacology
  • Aspirin / therapeutic use
  • Blood Platelets / drug effects
  • Blood Platelets / pathology
  • CD8-Positive T-Lymphocytes / pathology
  • Carcinoma, Hepatocellular / pathology
  • Carcinoma, Hepatocellular / prevention & control*
  • Carcinoma, Hepatocellular / virology*
  • Cell Proliferation / drug effects
  • Clopidogrel
  • Disease Models, Animal
  • Hepatitis B virus*
  • Hepatitis B, Chronic / complications*
  • Hepatitis B, Chronic / pathology
  • Humans
  • Liver Neoplasms / pathology
  • Liver Neoplasms / prevention & control*
  • Liver Neoplasms / virology*
  • Mice
  • Platelet Aggregation Inhibitors / pharmacology
  • Platelet Aggregation Inhibitors / therapeutic use*
  • Ticlopidine / analogs & derivatives
  • Ticlopidine / pharmacology
  • Ticlopidine / therapeutic use

Substances

  • Platelet Aggregation Inhibitors
  • Clopidogrel
  • Ticlopidine
  • Aspirin