The insulin-like growth factor II receptor is phosphorylated by a tyrosine kinase in adipocyte plasma membranes

J Biol Chem. 1986 Jun 15;261(17):7675-9.

Abstract

Incorporation of 32P from [gamma-32P]ATP into tyrosine residues of the insulin-like growth factor (IGF)-II receptor was observed in a Triton X-100-insoluble fraction of rat adipocyte plasma membranes. IGF-II receptor phosphorylation proceeded to a stoichiometry of approximately 0.5 mol of phosphate/IGF-II binding site after 10 min of incubation at 4 degrees C. A Km for ATP of 6 microM was calculated for this phosphorylation reaction. Addition of IGF-II caused an approximately 2-fold increase in tyrosine phosphorylation of the IGF-II receptor in this preparation. In contrast, phosphorylation of angiotensin II by the Triton X-100 washed membranes was not stimulated by IGF-II. Incubation of purified receptor immobilized on IGF-II agarose or of receptor-enriched low density microsomal membranes with [gamma-32P]ATP did not result in appreciable incorporation of [32P]phosphate into the IGF-II receptor nor into exogenous substrates. These data suggest that the IGF-II receptor is not a tyrosine protein kinase capable of autophosphorylation but that it is a substrate for a tyrosine protein kinase endogenous to the adipocyte plasma membrane. The stimulatory effect of IGF-II on the tyrosine phosphorylation of its receptor may be due to a conformational change which converts the receptor to a better substrate for this tyrosine kinase.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adenosine Triphosphate / metabolism
  • Adipose Tissue / enzymology
  • Adipose Tissue / metabolism*
  • Angiotensin II / metabolism
  • Animals
  • Cell Membrane / enzymology
  • Insulin-Like Growth Factor II / metabolism*
  • Kinetics
  • Male
  • Molecular Weight
  • Phosphorus Radioisotopes
  • Phosphotyrosine
  • Protein-Tyrosine Kinases / metabolism*
  • Rats
  • Rats, Inbred Strains
  • Receptors, Cell Surface / isolation & purification
  • Receptors, Cell Surface / metabolism*
  • Receptors, Somatomedin
  • Somatomedins / metabolism*
  • Tyrosine / analogs & derivatives
  • Tyrosine / analysis

Substances

  • Phosphorus Radioisotopes
  • Receptors, Cell Surface
  • Receptors, Somatomedin
  • Somatomedins
  • Angiotensin II
  • Phosphotyrosine
  • Tyrosine
  • Insulin-Like Growth Factor II
  • Adenosine Triphosphate
  • Protein-Tyrosine Kinases