Synthesis, characterization, controlled release, and antibacterial studies of a novel streptomycin chitosan magnetic nanoantibiotic

Int J Nanomedicine. 2014 Jan 16:9:549-57. doi: 10.2147/IJN.S53079. eCollection 2014.

Abstract

This study describes the preparation, characterization, and controlled release of a streptomycin-chitosan-magnetic nanoparticle-based antibiotic in an effort to improve the treatment of bacterial infections. Specifically, chitosan-magnetic nanoparticles were synthesized by an incorporation method and were characterized by Fourier transform infrared spectroscopy, X-ray diffraction, thermogravimetric analysis, and vibrating sample magnetometry. Streptomycin was incorporated into the nanoparticles to form a streptomycin-coated chitosan-magnetic nanoparticle (Strep-CS-MNP) nanocomposite. The release profiles showed an initially fast release, which became slower as time progressed. The percentage of drug released after 350 minutes was around 100%, and the best fit mathematical model for drug release was the pseudo-second order model. The Strep-CS-MNP nanocomposite showed enhanced antibacterial activity against methicillin-resistant Staphylococcus aureus. This study forms a significant basis for further investigation of the Strep-CS-MNP nanocomposite in the treatment of various bacterial infections.

Keywords: antimicrobial activity; chitosan; magnetic nanoparticles; methicillin-resistant Staphylococcus aureus; nanoantibiotics; release; streptomycin.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Anti-Bacterial Agents / administration & dosage*
  • Anti-Bacterial Agents / pharmacokinetics
  • Chitosan / chemistry*
  • Delayed-Action Preparations
  • Humans
  • Magnetite Nanoparticles / administration & dosage*
  • Magnetite Nanoparticles / chemistry*
  • Magnetite Nanoparticles / ultrastructure
  • Methicillin-Resistant Staphylococcus aureus / drug effects
  • Microbial Sensitivity Tests
  • Models, Biological
  • Molecular Structure
  • Nanocomposites / administration & dosage
  • Nanocomposites / chemistry
  • Nanocomposites / ultrastructure
  • Nanomedicine
  • Spectroscopy, Fourier Transform Infrared
  • Streptomycin / administration & dosage*
  • Streptomycin / pharmacokinetics
  • X-Ray Diffraction

Substances

  • Anti-Bacterial Agents
  • Delayed-Action Preparations
  • Magnetite Nanoparticles
  • Chitosan
  • Streptomycin