Albendazolesulphoxide concentrations in plasma and hydatid cyst and prediction of parasitological and clinical outcomes in patients with liver hydatidosis caused by Echinococcus granulosus

Croat Med J. 2014 Apr;55(2):146-55. doi: 10.3325/cmj.2014.55.146.

Abstract

Aim: To investigate the relationship between plasma and cyst concentrations of albendazolesulphoxide (ASO) and their effects on parasitological findings and disease recurrence in patients with liver hydatidosis.

Methods: The study was conducted at the University Hospital for Infectious Diseases Dr. Fran Mihaljević, Zagreb, Croatia, between August 2006 and January 2011. Consecutive patients (N=48, age 6-77 years) were treated with albendazole (3×5 mg/kg/d) over 28 days before surgical cyst removal (n=34) or percutaneous evacuation (PAIR) (n=14). Plasma ASO was determined on days 10 and 28 of treatment and cyst concentrations at surgery/PAIR.

Results: Disease recurred in 3 surgically treated patients. Variability of ASO concentrations was substantial. Plasma concentrations on day 10 were higher than on day 28 (geometric means ratio [GMR] 2.00; 95%CI 1.38-2.91, P<0.001) and higher than cyst concentrations at the time of treatment (GMR=1.58, 1.01-2.34, P=0.045). Higher cyst (but not plasma) concentrations were independently associated with lower odds of protoscolex motility (OR=0.23, 0.01-0.70, P<0.001) and higher odds of protoscolex destruction (OR=1.17, 1.04-1.46, P<0.001). With adjustment for age and protoscolex motility, higher day 10 plasma concentrations (but not cyst concentrations) were associated with lower odds of disease recurrence (OR=0.49, 0.09-0.97, P=0.035). Plasma concentrations did not predict cyst concentrations.

Conclusion: Viability of protoscolices progressively decreased with increasing ASO concentrations in the cyst. Data strongly suggested that higher plasma concentrations reduced the risk of disease recurrence.

MeSH terms

  • Adolescent
  • Adult
  • Aged
  • Albendazole / analogs & derivatives*
  • Albendazole / pharmacokinetics
  • Animals
  • Anthelmintics / pharmacokinetics*
  • Antibodies, Helminth / blood
  • Antigens, Helminth / immunology
  • Biological Availability
  • Child
  • Echinococcosis, Hepatic / diagnosis
  • Echinococcosis, Hepatic / drug therapy
  • Echinococcosis, Hepatic / metabolism*
  • Echinococcosis, Hepatic / surgery
  • Echinococcus granulosus / drug effects*
  • Echinococcus granulosus / immunology
  • Enzyme-Linked Immunosorbent Assay
  • Female
  • Humans
  • Male
  • Middle Aged
  • Recurrence
  • Treatment Outcome
  • Young Adult

Substances

  • Anthelmintics
  • Antibodies, Helminth
  • Antigens, Helminth
  • Albendazole
  • albendazole sulfoxide