Therapeutic targets in subependymoma

J Neuroimmunol. 2014 Dec 15;277(1-2):168-75. doi: 10.1016/j.jneuroim.2014.10.008. Epub 2014 Oct 31.

Abstract

Subependymomas are usually treated with surgical resection; however, no standard, defined alternative medical therapy is recommended for patients who are not surgical candidates, owing to a paucity of molecular, immunological, and genetic characterization. To address this, an ex vivo functional analysis of the immune microenvironment in subependymoma was conducted, a subependymoma cytokine/chemokine microarray was constructed for the evaluation of operational immune and molecular pathways, and a subependymoma cell line was derived and used to test a variety of cytotoxic agents that target operational pathways identified in subependymoma. We found that immune effectors are detectable within the microenvironment of subependymoma; however, marked immune suppression is not observed. The subependymoma tissue microarrays demonstrated tumor expression of p53, MDM2, HIF-1α, topoisomerase II-β, p-STAT3, and nucleolin, but not EGFRvIII, EphA2, IL-13RA2, CMV, CTLA-4, FoxP3, PD-1, PD-L1, EGFR, PDGF-α, PDGF-β, PDGFR-α, PDGFR-β, PTEN, IGFBP2, PI3K, MDM4, IDH1, mTOR, or Jak2. A topoisomerase inhibitor (WP744, IC50=0.83 μM) and a p-STAT3/HIF-1α inhibitor (WP1066, IC50=3.15 μM) demonstrated a growth inhibition of the subependymoma cell proliferation. Cumulatively, these data suggest that those agents that interfere with oncogenes operational in subependymoma may have clinical impact.

Keywords: Ependymoma; Immunotherapy; Noninvasive; Subependymoma.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antineoplastic Agents / chemistry
  • Antineoplastic Agents / pharmacology
  • Antineoplastic Agents / therapeutic use
  • Brain Neoplasms / embryology
  • Brain Neoplasms / metabolism
  • Brain Neoplasms / pathology*
  • Cell Line, Tumor / drug effects
  • Cell Proliferation / drug effects
  • Colony-Forming Units Assay
  • Cytokines / genetics
  • Cytokines / metabolism
  • Cytotoxicity Tests, Immunologic
  • Dose-Response Relationship, Drug
  • Drug Screening Assays, Antitumor*
  • Flow Cytometry
  • Gene Expression Regulation, Neoplastic / drug effects
  • Glioma, Subependymal / immunology
  • Glioma, Subependymal / metabolism
  • Glioma, Subependymal / pathology*
  • Humans
  • Neoplasm Proteins / genetics
  • Neoplasm Proteins / metabolism*
  • Neoplastic Stem Cells / drug effects
  • Neoplastic Stem Cells / immunology
  • Neoplastic Stem Cells / metabolism
  • Pyridines / chemistry
  • Pyridines / pharmacology
  • Signal Transduction / drug effects
  • Signal Transduction / physiology
  • T-Lymphocytes / drug effects
  • T-Lymphocytes / immunology
  • Tissue Array Analysis
  • Tyrphostins / chemistry
  • Tyrphostins / pharmacology

Substances

  • Antineoplastic Agents
  • Cytokines
  • Neoplasm Proteins
  • Pyridines
  • Tyrphostins
  • WP1066