Anomalous oxidative cleavage of the side chain of 18-oxocortisol and its tetrahydro metabolite

J Steroid Biochem. 1989 Oct;33(4A):605-11. doi: 10.1016/0022-4731(89)90048-4.

Abstract

The course of oxidative side chain cleavage of two recently isolated 17 alpha-hydroxy C-18 oxygenated naturally-occurring corticosteroids differed in that 18-hydroxycortisol yielded a 17-ketosteroid (Chu M. D., and Ulick S. (1982) J. biol. Chem. 257, 2218-2224) whereas 18-oxocortisol yielded a gamma-etiolactone (Ulick S., Chu M. D. and Land M. (1983) J. biol. Chem. 258, 5498-5502). In an analytic application of the periodic acid oxidative cleavage reaction to 18-oxocortisol, the finding of a second product of the reaction prompted a reinvestigation of its course. Both the delta 4,3-ketone secreted form of the steroid and its tetrahydro urinary metabolite were cleaved predominantly to 17-ketosteroids along with smaller amounts of gamma-etiolactones, whose proof of structure is herein reported. This anomalous course of oxidative cleavage was considered to reflect an equilibrium between C-20 ketone and cyclic-hemiketal forms in which the glycerol-type side chain structure of the later becomes the precursor of a 17-ketosteroid. Because of the similarities between in vitro oxidative side chain cleavage and in vivo corticosteroid metabolism, these findings suggest that C-18 oxygenated steroids may contribute to the 17-ketosteroid fraction of human urine.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Gas Chromatography-Mass Spectrometry
  • Hydrocortisone / analogs & derivatives*
  • Hydrocortisone / metabolism
  • Ketosteroids / metabolism
  • Lactones / metabolism
  • Oxidation-Reduction
  • Periodic Acid
  • Trimethylsilyl Compounds / metabolism

Substances

  • Ketosteroids
  • Lactones
  • Trimethylsilyl Compounds
  • Periodic Acid
  • 18-oxocortisol
  • Hydrocortisone