[3H]PN200-110 and [3H]ryanodine binding and reconstitution of ion channel activity with skeletal muscle membranes

Anal Biochem. 1989 Nov 15;183(1):31-41. doi: 10.1016/0003-2697(89)90167-x.

Abstract

Skeletal muscle membranes derived either from the tubular (T) network or from the sarcoplasmic reticulum (SR) were characterized with respect to the binding of the dihydropyridine, [3H]PN200-110, and the alkaloid, [3H]ryanodine; polypeptide composition; and ion channel activity. Conditions for optimizing the binding of these radioligands are discussed. A bilayer pulsing technique is described and is used to examine the channels present in these membranes. Fusion of T-tubule membranes into bilayers revealed the presence of chloride channels and dihydropyridine-sensitive calcium channels with three distinct conductances. The dihydropyridine-sensitive channels were further characterized with respect to their voltage dependence. Pulsing experiments indicated that two different populations of dihydropyridine-sensitive channels existed. Fusion of heavy SR vesicles revealed three different ion channels; the putative calcium release channel, a potassium channel, and a chloride channel. Thus, this fractionation procedure provides T-tubules and SR membranes which, with radioligand binding and single channel recording techniques, provide a useful tool to study the characteristics of skeletal muscle ion channels and their possible role in excitation-contraction coupling.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Alkaloids / metabolism*
  • Animals
  • Calcium Channel Blockers / metabolism*
  • Calcium Channels / physiology
  • Chloride Channels
  • Chlorides / metabolism
  • Dihydropyridines / pharmacology
  • Electrophoresis / methods
  • Isradipine
  • Lipid Bilayers / metabolism
  • Membrane Proteins / metabolism
  • Membranes / metabolism
  • Muscles / metabolism*
  • Oxadiazoles / metabolism*
  • Potassium Channels / physiology
  • Rabbits
  • Ryanodine / metabolism*
  • Sarcoplasmic Reticulum / ultrastructure
  • Tritium

Substances

  • Alkaloids
  • Calcium Channel Blockers
  • Calcium Channels
  • Chloride Channels
  • Chlorides
  • Dihydropyridines
  • Lipid Bilayers
  • Membrane Proteins
  • Oxadiazoles
  • Potassium Channels
  • Tritium
  • Ryanodine
  • 1,4-dihydropyridine
  • Isradipine