Effect of Culture Conditions on Metabolite Production of Xylaria sp

Molecules. 2015 Apr 30;20(5):7940-50. doi: 10.3390/molecules20057940.

Abstract

Seeking a strategy for triggering the cryptic natural product biosynthesis to yield novel compounds in the plant-associated fungus Xylaria sp., the effect of culture conditions on metabolite production was investigated. A shift in the production of five known cytochalasin-type analogues 1-5 to six new α-pyrone derivatives, xylapyrones A-F (compounds 6-11), from a solid to a liquid medium was observed. These compounds were identified by analysis of 1D and 2D NMR and HRMS data. Compounds 1-3 showed moderate cytotoxicity against HepG2 and Caski cancer cell lines with IC50 values ranging from 25 to 63 μM and compounds 4-11 were found to be inactive, with IC50 values>100 μM.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Biological Products / chemistry*
  • Biological Products / metabolism*
  • Cell Culture Techniques / methods
  • Cell Line, Tumor
  • Cytochalasins / chemistry*
  • Cytochalasins / metabolism*
  • Hep G2 Cells
  • Humans
  • Magnetic Resonance Spectroscopy / methods
  • Xylariales / chemistry*
  • Xylariales / metabolism*

Substances

  • Biological Products
  • Cytochalasins