Belinostat for the treatment of relapsed or refractory peripheral T-cell lymphoma

Future Oncol. 2015;11(11):1659-64. doi: 10.2217/fon.15.62.

Abstract

The prognosis of patients with relapsed/refractory peripheral T-cell lymphoma (PTCL) remains poor and current treatments are typically of limited benefit. Histone deacetylase (HDAC) inhibitors have proven effective for the treatment of relapsed/refractory PTCL. To date approved HDAC inhibitors for patients with T-cell lymphoma are vorinostat, romidepsin and, recently, belinostat. Here we review the pharmacology and the clinical activity of belinostat. Belinostat is a well-tolerated HDAC inhibitor that has shown activity in heavily pretreated patients with relapsed/refractory PTCL. Several clinical trials are currently investigating the use of belinostat in different cancers and in combination with other chemotherapeutic agents.

Keywords: T-cell lymphoma; belinostat; histone deacetylase inhibitor.

Publication types

  • Review

MeSH terms

  • Antineoplastic Agents / chemistry
  • Antineoplastic Agents / therapeutic use*
  • Clinical Trials as Topic
  • Humans
  • Hydroxamic Acids / chemistry
  • Hydroxamic Acids / therapeutic use*
  • Lymphoma, T-Cell, Peripheral / drug therapy*
  • Recurrence
  • Retreatment
  • Sulfonamides / chemistry
  • Sulfonamides / therapeutic use*

Substances

  • Antineoplastic Agents
  • Hydroxamic Acids
  • Sulfonamides
  • belinostat