New compounds, nanaomycin F and G, discovered by physicochemical screening from a culture broth of Streptomyces rosa subsp. notoensis OS-3966

J Biosci Bioeng. 2015 Nov;120(5):596-600. doi: 10.1016/j.jbiosc.2015.03.018. Epub 2015 Jun 20.

Abstract

Two new compounds, nanaomycin F and G, were isolated by physicochemical screening method from cultured broth of Streptomyces rosa subsp. notoensis OS-3966, which is known to produce nanaomycin A, B, C, D, and E. Nanaomycin F is a new nanaomycin analog, a 4a-hydroxyl analog of nanaomycin B. Nanaomycin G has a unique skeleton with 1-indanone infused with a tetrahydropyran ring. Nanaomycin A possesses broad antimicrobial activity but nanaomycin F and G demonstrated no bioactivity against all bacteria and fungi tested in this study. In addition, in both nanaomycin F and G, the production of superoxide radicals was majorly decreased in comparison to nanaomycin A. It was considered that the antimicrobial properties were lost as a result of the decrease in production of the superoxide radicals.

Keywords: Nanaomycin F; Nanaomycin G; Nanaomycin analogs; Physicochemical screening; Streptomyces sp..

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Anti-Bacterial Agents / chemistry
  • Anti-Bacterial Agents / isolation & purification
  • Anti-Bacterial Agents / pharmacology
  • Antifungal Agents / chemistry
  • Antifungal Agents / isolation & purification
  • Antifungal Agents / pharmacology
  • Bacteria / drug effects
  • Fungi / drug effects
  • Hydroxylation
  • Indans / chemistry
  • Naphthoquinones / chemistry*
  • Naphthoquinones / isolation & purification*
  • Naphthoquinones / pharmacology
  • Streptomyces / chemistry*
  • Streptomyces / growth & development
  • Superoxides / metabolism

Substances

  • Anti-Bacterial Agents
  • Antifungal Agents
  • Indans
  • Naphthoquinones
  • nanaomycin F
  • nanaomycin G
  • Superoxides
  • nanaomycin A
  • nanaomycin B