Glucagon sensitivity and clearance in type 1 diabetes: insights from in vivo and in silico experiments

Am J Physiol Endocrinol Metab. 2015 Sep 1;309(5):E474-86. doi: 10.1152/ajpendo.00236.2015. Epub 2015 Jul 7.

Abstract

Glucagon use in artificial pancreas for type 1 diabetes (T1D) is being explored for prevention and rescue from hypoglycemia. However, the relationship between glucagon stimulation of endogenous glucose production (EGP) viz., hepatic glucagon sensitivity, and prevailing glucose concentrations has not been examined. To test the hypothesis that glucagon sensitivity is increased at hypoglycemia vs. euglycemia, we studied 29 subjects with T1D randomized to a hypoglycemia or euglycemia clamp. Each subject was studied at three glucagon doses at euglycemia or hypoglycemia, with EGP measured by isotope dilution technique. The peak EGP increments and the integrated EGP response increased with increasing glucagon dose during euglycemia and hypoglycemia. However, the difference in dose response based on glycemia was not significant despite higher catecholamine concentrations in the hypoglycemia group. Knowledge of glucagon's effects on EGP was used to develop an in silico glucagon action model. The model-derived output fitted the obtained data at both euglycemia and hypoglycemia for all glucagon doses tested. Glucagon clearance did not differ between glucagon doses studied in both groups. Therefore, the glucagon controller of a dual hormone control system may not need to adjust glucagon sensitivity, and hence glucagon dosing, based on glucose concentrations during euglycemia and hypoglycemia.

Keywords: endogenous glucose production; glucagon; type 1 diabetes.

Publication types

  • Randomized Controlled Trial
  • Research Support, N.I.H., Extramural

MeSH terms

  • Adult
  • Blood Glucose / drug effects
  • Blood Glucose / metabolism*
  • Computer Simulation
  • Diabetes Mellitus, Type 1 / metabolism*
  • Female
  • Glucagon / pharmacology*
  • Gluconeogenesis / drug effects*
  • Glucose / metabolism
  • Glucose Clamp Technique
  • Glycogenolysis / drug effects*
  • Hormones / pharmacology*
  • Humans
  • Hypoglycemia / metabolism*
  • Liver / drug effects*
  • Liver / metabolism
  • Male
  • Middle Aged
  • Pancreas, Artificial
  • Young Adult

Substances

  • Blood Glucose
  • Hormones
  • Glucagon
  • Glucose