Mathematical modeling reveals a critical role for cyclin D1 dynamics in phenotype switching during glioma differentiation

FEBS Lett. 2015 Aug 19;589(18):2304-11. doi: 10.1016/j.febslet.2015.07.014. Epub 2015 Jul 17.

Abstract

Glioma differentiation therapy is a novel modality to increase anti-glioma effects using specific drugs to induce glioma cell differentiation to glia-like cells. However, the molecular mechanisms underlying glioma differentiation remain poorly understood. In this study, we built an experiment-integrated mathematical model for glioma differentiation signaling pathways. Our modeling and experimental analysis revealed that a "one-way-switch" bifurcation of cyclin D1 dynamics was critical for controlling the phenotypic transition of glioma cells. We also quantitatively evaluated drug combinations toward a synergistic therapeutic effect. These results provide insights into the molecular mechanisms underlying glioma differentiation and implications for the design of novel therapeutic targets in anti-cancer therapy.

Keywords: Cyclin D1; Glioma differentiation; Mathematical modeling; Phenotype switching.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antineoplastic Agents / pharmacology
  • Cell Differentiation* / drug effects
  • Cell Line, Tumor
  • Cell Proliferation / drug effects
  • Cyclin D1 / metabolism*
  • Drug Synergism
  • Glioma / pathology*
  • Models, Biological*
  • Phenotype*
  • Rats
  • Signal Transduction / drug effects

Substances

  • Antineoplastic Agents
  • Cyclin D1