Polyethylenimine-coated SPION exhibits potential intrinsic anti-metastatic properties inhibiting migration and invasion of pancreatic tumor cells

J Control Release. 2015 Oct 28:216:78-92. doi: 10.1016/j.jconrel.2015.08.009. Epub 2015 Aug 8.

Abstract

Due to its aggressive behavior, pancreatic cancer is one of the principal causes of cancer-related deaths. The highly metastatic potential of pancreatic tumor cells demands the development of more effective anti-metastatic approaches for this disease. Although polyethylenimine-coated superparamagnetic iron oxide nanoparticles (PEI-coated SPIONs) have been studied for their utility as transfection agents, little is known of their effect on tumor cell biology. Here we demonstrated that PEI-coated SPIONs have potent inhibitory effects on pancreatic tumor cell migration/invasion, through inhibition of Src kinase and decreased expression of MT1-MMP and MMP2 metalloproteinases. When treated with PEI-coated SPIONs, the pancreatic tumor cell line Pan02 showed reduced invadosome density and thus, a decrease in their ability to invade through basement membrane. These nanoparticles temporarily downmodulated microRNA-21, thereby upregulating the cell migration inhibitors PTEN, PDCD4 and Sprouty-1. PEI-coated SPIONs thus show intrinsic, possibly anti-metastatic properties for modulating pancreatic tumor cell migration machinery, which indicates their potential as anti-metastatic agents for treatment of pancreatic cancer.

Keywords: Matrix degradation; Nanoparticle; Proliferation; Tumor cell invasion; Tumor cell migration.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cell Line, Tumor
  • Cell Movement / drug effects
  • Cell Movement / genetics
  • Cell Proliferation / drug effects
  • Ferric Compounds / chemistry*
  • Ferric Compounds / therapeutic use*
  • Gene Transfer Techniques*
  • HEK293 Cells
  • Humans
  • Magnetics
  • Matrix Metalloproteinase Inhibitors / pharmacology
  • MicroRNAs
  • Nanoparticles
  • Neoplasm Invasiveness
  • Neoplasm Metastasis / therapy*
  • Pancreatic Neoplasms / drug therapy*
  • Polyethyleneimine / chemistry*
  • Signal Transduction / drug effects
  • Transfection

Substances

  • Ferric Compounds
  • MIRN21 microRNA, human
  • Matrix Metalloproteinase Inhibitors
  • MicroRNAs
  • ferric oxide
  • Polyethyleneimine