A Novel Compound Analgesic Cream (Ketamine, Pentoxifylline, Clonidine, DMSO) for Complex Regional Pain Syndrome Patients

Pain Pract. 2016 Jan;16(1):E14-20. doi: 10.1111/papr.12404. Epub 2015 Nov 7.

Abstract

Background: Evidence suggests that complex regional pain syndrome (CRPS) is a manifestation of microvascular dysfunction. Topical combinations of α2-adrenergic receptor agonists or nitric oxide donors with phosphodiesterase or phosphatidic acid inhibitors formulated to treat microvascular dysfunction have been shown to reduce allodynia in a rat model of CRPS-I. Driven by these findings, we assessed the outcomes of CRPS patients treated with a compound analgesic cream (CAC) consisting of ketamine 10%, pentoxifylline 6%, clonidine 0.2%, and dimethyl sulfoxide 6% to 10%.

Methods: An audit was conducted on 13 CRPS patients who trialed the CAC. A detailed report was compiled for each patient which comprised baseline characteristics, including CRPS description, previous treatments, and pain scores (numerical pain rating scale; 0 to 10). Recorded outcomes consisted of pain scores, descriptive outcomes, and concurrent medications/treatments, for which basic analysis was performed to determine the effectiveness of the CAC. Case reports are presented for 3 patients with varying outcomes.

Results: Nine patients (69%) reported pain/symptom reduction (4.4 ± 2.1 vs. 6.3 ± 1.9) with use of the CAC. Six patients reported sustained benefits after 2 months of CAC use, and 2 patients reported complete resolution of pain/symptoms: one had early CRPS-I and the other received a partial CRPS diagnosis. An otherwise medication refractory and intolerant patient found partial benefit with the CAC.

Conclusions: These results demonstrate promise for this topical combination as a useful treatment in multimodal therapy for patients with CRPS, with the potential to resolve pain/symptoms in early CRPS patients.

Keywords: NO donor; clonidine; complex regional pain syndrome; dimethyl sulfoxide; ketamine; nitric oxide complex regional pain syndrome; pentoxifylline; topical analgesic.

Publication types

  • Case Reports

MeSH terms

  • Adrenergic alpha-Agonists / administration & dosage*
  • Adrenergic alpha-Agonists / adverse effects
  • Adrenergic alpha-Agonists / therapeutic use*
  • Adult
  • Analgesics / administration & dosage*
  • Analgesics / therapeutic use*
  • Anesthetics, Dissociative / administration & dosage*
  • Anesthetics, Dissociative / adverse effects
  • Anesthetics, Dissociative / therapeutic use*
  • Anti-Infective Agents, Local / administration & dosage*
  • Anti-Infective Agents, Local / adverse effects
  • Anti-Infective Agents, Local / therapeutic use*
  • Causalgia / drug therapy
  • Clonidine / administration & dosage*
  • Clonidine / adverse effects
  • Clonidine / therapeutic use*
  • Complex Regional Pain Syndromes / drug therapy*
  • Dimethyl Sulfoxide / administration & dosage*
  • Dimethyl Sulfoxide / adverse effects
  • Dimethyl Sulfoxide / therapeutic use*
  • Female
  • Humans
  • Ketamine / administration & dosage*
  • Ketamine / adverse effects
  • Ketamine / therapeutic use*
  • Male
  • Middle Aged
  • Ointments
  • Pain Measurement
  • Pentoxifylline / administration & dosage*
  • Pentoxifylline / adverse effects
  • Pentoxifylline / therapeutic use*
  • Phosphodiesterase Inhibitors / administration & dosage*
  • Phosphodiesterase Inhibitors / adverse effects
  • Phosphodiesterase Inhibitors / therapeutic use*
  • Reflex Sympathetic Dystrophy / drug therapy
  • Treatment Outcome

Substances

  • Adrenergic alpha-Agonists
  • Analgesics
  • Anesthetics, Dissociative
  • Anti-Infective Agents, Local
  • Ointments
  • Phosphodiesterase Inhibitors
  • Ketamine
  • Clonidine
  • Pentoxifylline
  • Dimethyl Sulfoxide