Pharmacokinetics and Clinical Utility of Valproic Acid Administered via Continuous Infusion

CNS Drugs. 2016 Jan;30(1):71-7. doi: 10.1007/s40263-015-0304-5.

Abstract

Introduction: Valproic acid is a versatile antiepileptic drug that is often used in the acute care setting. Intravenous valproic acid lends itself well to a continuous infusion as it exhibits a relatively short half-life. We evaluated the pharmacokinetics and clinical efficacy of continuous infusion valproic acid in hospitalized patients with migraine and seizures.

Methods: A retrospective cohort study was performed utilizing information from the medical records of patients receiving an intravenous continuous infusion of valproic acid. Patients were included if they were aged 1 month to 85 years and they received a continuous infusion of valproic acid. Therapeutic response, common adverse effects, and the pharmacokinetic profile of valproic acid were evaluated.

Results: Continuous infusion valproic acid led to a concentration within the desired range (50-100 μg/ml) in 83.4% of patients, a rate that was higher in pediatric patients. The clinical response rate was also higher in pediatric patients with seizures or migraines and appeared to be better when the concentration was >75 μg/ml. Analysis of safety parameters suggests similar safety considerations to valproic acid when administered via intermittent infusion.

Conclusions: Continuous infusion valproic acid appears to be a safe, effective, and predictable manner by which to administer valproic acid to pediatric and adult patients admitted to the hospital.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Adolescent
  • Adult
  • Aged
  • Aged, 80 and over
  • Anticonvulsants / administration & dosage*
  • Anticonvulsants / adverse effects
  • Anticonvulsants / blood*
  • Anticonvulsants / therapeutic use
  • Child
  • Child, Preschool
  • Cohort Studies
  • Data Interpretation, Statistical
  • Female
  • Humans
  • Infant
  • Infusions, Intravenous
  • Male
  • Medical Records
  • Middle Aged
  • Migraine Disorders / drug therapy
  • Retrospective Studies
  • Seizures / drug therapy
  • Treatment Outcome
  • Valproic Acid / administration & dosage*
  • Valproic Acid / adverse effects
  • Valproic Acid / blood*
  • Valproic Acid / therapeutic use
  • Young Adult

Substances

  • Anticonvulsants
  • Valproic Acid