Agomelatine Increases BDNF Serum Levels in Depressed Patients in Correlation with the Improvement of Depressive Symptoms

Int J Neuropsychopharmacol. 2016 Apr 29;19(5):pyw003. doi: 10.1093/ijnp/pyw003. Print 2016 May.

Abstract

Background: Agomelatine modulates brain-derived neurotrophic factor expression via its interaction with melatonergic and serotonergic receptors and has shown promising results in terms of brain-derived neurotrophic factor increase in animal models.

Methods: Twenty-seven patients were started on agomelatine (25mg/d). Venous blood was collected and brain-derived neurotrophic factor serum levels were measured at baseline and after 2 and 8 weeks along with a clinical assessment, including Hamilton Depression Rating Scale and Snaith-Hamilton Pleasure Scale.

Results: Brain-derived neurotrophic factor serum concentration increased after agomelatine treatment. Responders showed a significant increase in brain-derived neurotrophic factor levels after 2 weeks of agomelatine treatment; no difference was observed in nonresponders. Linear regression analysis showed that more prominent brain-derived neurotrophic factor level variation was associated with lower baseline BDNF levels and greater anhedonic features at baseline.

Conclusions: Patients affected by depressive disorders showed an increase of brain-derived neurotrophic factor serum concentration after a 2-week treatment with agomelatine. The increase of brain-derived neurotrophic factor levels was found to be greater in patients with lower brain-derived neurotrophic factor levels and marked anhedonia at baseline.

Keywords: BDNF; agomelatine; major depressive disorder.

Publication types

  • Randomized Controlled Trial

MeSH terms

  • Acetamides / therapeutic use*
  • Affect / drug effects*
  • Aged
  • Antidepressive Agents / therapeutic use*
  • Biomarkers / blood
  • Brain-Derived Neurotrophic Factor / blood*
  • Depression / blood
  • Depression / diagnosis
  • Depression / drug therapy*
  • Depression / psychology
  • Female
  • Humans
  • Italy
  • Linear Models
  • Male
  • Middle Aged
  • Remission Induction
  • Time Factors
  • Treatment Outcome
  • Up-Regulation

Substances

  • Acetamides
  • Antidepressive Agents
  • Biomarkers
  • Brain-Derived Neurotrophic Factor
  • agomelatine
  • BDNF protein, human