Ibrutinib enhances chimeric antigen receptor T-cell engraftment and efficacy in leukemia

Blood. 2016 Mar 3;127(9):1117-27. doi: 10.1182/blood-2015-11-679134. Epub 2016 Jan 26.

Abstract

Anti-CD19 chimeric antigen receptor (CAR) T-cell therapy is highly promising but requires robust T-cell expansion and engraftment. A T-cell defect in chronic lymphocytic leukemia (CLL) due to disease and/or therapy impairs ex vivo expansion and response to CAR T cells. To evaluate the effect of ibrutinib treatment on the T-cell compartment in CLL as it relates to CAR T-cell generation, we examined the phenotype and function of T cells in a cohort of CLL patients during their course of treatment with ibrutinib. We found that ≥5 cycles of ibrutinib therapy improved the expansion of CD19-directed CAR T cells (CTL019), in association with decreased expression of the immunosuppressive molecule programmed cell death 1 on T cells and of CD200 on B-CLL cells. In support of these findings, we observed that 3 CLL patients who had been treated with ibrutinib for ≥1 year at the time of T-cell collection had improved ex vivo and in vivo CTL019 expansion, which correlated positively together and with clinical response. Lastly, we show that ibrutinib exposure does not impair CAR T-cell function in vitro but does improve CAR T-cell engraftment, tumor clearance, and survival in human xenograft models of resistant acute lymphocytic leukemia and CLL when administered concurrently. Our collective findings indicate that ibrutinib enhances CAR T-cell function and suggest that clinical trials with combination therapy are warranted. Our studies demonstrate that improved T-cell function may also contribute to the efficacy of ibrutinib in CLL. These trials were registered at www.clinicaltrials.gov as #NCT01747486, #NCT01105247, and #NCT01217749.

Publication types

  • Clinical Trial
  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenine / analogs & derivatives
  • Administration, Oral
  • Aged
  • Animals
  • Antigens, CD / metabolism
  • Cell Line, Tumor
  • Cell Proliferation / drug effects
  • Cytotoxicity, Immunologic / drug effects
  • Demography
  • Disease Models, Animal
  • Drug Resistance, Neoplasm / drug effects
  • Gene Transfer Techniques
  • Humans
  • Immunosuppression Therapy
  • K562 Cells
  • Leukemia, Lymphocytic, Chronic, B-Cell / drug therapy*
  • Leukemia, Lymphocytic, Chronic, B-Cell / immunology*
  • Leukemia, Lymphocytic, Chronic, B-Cell / pathology
  • Male
  • Mice
  • Middle Aged
  • Piperidines
  • Programmed Cell Death 1 Receptor / metabolism
  • Pyrazoles / administration & dosage
  • Pyrazoles / pharmacology
  • Pyrazoles / therapeutic use*
  • Pyrimidines / administration & dosage
  • Pyrimidines / pharmacology
  • Pyrimidines / therapeutic use*
  • Receptors, Antigen, T-Cell / metabolism*
  • T-Lymphocytes / drug effects
  • T-Lymphocytes / immunology*
  • Time Factors
  • Treatment Outcome

Substances

  • Antigens, CD
  • CTL019 chimeric antigen receptor
  • PDCD1 protein, human
  • Piperidines
  • Programmed Cell Death 1 Receptor
  • Pyrazoles
  • Pyrimidines
  • Receptors, Antigen, T-Cell
  • ibrutinib
  • Adenine
  • antigens, CD200

Associated data

  • ClinicalTrials.gov/NCT01105247
  • ClinicalTrials.gov/NCT01217749
  • ClinicalTrials.gov/NCT01747486