Composition and biological activities of the essential oil of Piper corcovadensis (Miq.) C. DC (Piperaceae)

Exp Parasitol. 2016 Jun:165:64-70. doi: 10.1016/j.exppara.2016.03.017. Epub 2016 Mar 16.

Abstract

Essential oil from fresh leaves of the shrub Piper corcovadensis (Miq.) C. DC was obtained in 0.21% (w/w) yield by hydrodistillation in a Clevenger type apparatus. Thirty-one components, accounting for 96.61% of the leaf oil, were identified by gas chromatography-mass spectrometry. The major constituents of the oil were 1-butyl-3,4-methylenedioxybenzene (30.62%), terpinolene (17.44%), trans -caryophyllene (6.27%), α-pinene (5.92%), δ-cadinene (4.92%), and Limonene (4.46%). Bioassays against larvae of the Dengue mosquito (Aedes aegypti) revealed that leaf oil (LC50 = 30.52 ppm), terpinolene (LC50 = 31.16 ppm), and pure 1-butyl-3,4-methylenedioxybenzene (LC50 = 22.1 ppm) possessed larvicidal activities and are able to interfere with the activity of proteases from L4 gut enzymes. Additionally, the essential oil exhibited a strong oviposition deterrent activity at 50 and 5 ppm. This paper constitutes the first report of biological activities associated with the essential oil of leaves of P. corcovadensis.

Keywords: 1-Butyl-3,4-methylenedioxybenzene; Essential oil; Larvicidal activity; Oviposition activity; Piper corcovadensis; Piperaceae; Proteases enzymes.

MeSH terms

  • Aedes* / drug effects
  • Aedes* / physiology
  • Animals
  • Bicyclic Monoterpenes
  • Biological Assay
  • Cyclohexane Monoterpenes
  • Cyclohexenes / analysis
  • Dengue / transmission
  • Electrophoresis, Polyacrylamide Gel
  • Gas Chromatography-Mass Spectrometry
  • Larva / enzymology
  • Limonene
  • Monoterpenes / analysis
  • Mosquito Vectors* / drug effects
  • Mosquito Vectors* / physiology
  • Oils, Volatile / chemistry*
  • Oils, Volatile / isolation & purification
  • Oils, Volatile / pharmacology
  • Oviposition / drug effects
  • Peptide Hydrolases / analysis
  • Piper / chemistry*
  • Plant Leaves / chemistry
  • Polycyclic Sesquiterpenes
  • Protease Inhibitors / pharmacology
  • Sesquiterpenes / analysis
  • Terpenes / analysis
  • Trypsin / drug effects
  • Trypsin / metabolism

Substances

  • Bicyclic Monoterpenes
  • Cyclohexane Monoterpenes
  • Cyclohexenes
  • Monoterpenes
  • Oils, Volatile
  • Polycyclic Sesquiterpenes
  • Protease Inhibitors
  • Sesquiterpenes
  • Terpenes
  • delta-cadinene
  • Limonene
  • caryophyllene
  • Peptide Hydrolases
  • Trypsin
  • alpha-pinene
  • terpinolene